SCHEMBL8686333

SCHEMBL8686333

CN1CCC(c2c[nH]c3ccc(-c4ccsc4)cc23)C1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.57
ATM Q13315 1/20 0.57
HTR1D P28221 4/20 0.52
HTR1B P28222 4/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
THPO P40225 1/20 0.52
NOS3 P29474 4/20 0.52
NOS1 P29475 4/20 0.52
APP P05067 1/20 0.47
HTR1A P08908 1/20 0.46
HTR1F P30939 1/20 0.46
MAPT P10636 1/20 0.45
BLM P54132 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
GABRP O00591 1/20 0.45
GABRD O14764 1/20 0.45
GABRA1 P14867 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8686957 0.81 NOS3 (0.61) KDM4EATMHTR1DHTR1BCYP1A2
SCHEMBL8097614 0.81 KDM4E (0.58) KDM4EATMHTR1DHTR1BCYP1A2
SCHEMBL8508491 0.78 KDM4E (0.68) KDM4EATMHTR1DHTR1BCYP1A2
SCHEMBL8784248 0.77 KDM4E (0.57) KDM4EATMHTR1DHTR1BCYP1A2
SCHEMBL30877857 0.77 KDM4E (0.67) KDM4EATMHTR1DHTR1BCYP1A2
SCHEMBL29206549 0.77 KDM4E (0.67) KDM4EATMHTR1DHTR1BCYP1A2
SCHEMBL1122547 0.77 HTR1D (0.85) KDM4EATMHTR1DHTR1BCYP1A2
SCHEMBL2926854 0.77 KDM4E (0.67) KDM4EATMHTR1DHTR1BCYP1A2
SCHEMBL8474262 0.76 KDM4E (0.56) KDM4EATMHTR1DHTR1BCYP1A2
SCHEMBL7335724 0.76 HTR6 (0.68) KDM4EATMHTR1DHTR1BCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5770742-A SEROTONIN RECEPTOR SELECTIVITY, MIGRAINES ALLELIX BIOPHARMACEUTICALS INC. (CA) 1998-06-23 US claimed
WO-1997043281-A1 THIOPHENE- AND FURAN-TRYPTAMINE DERIVATIVES ALLELIX BIOPHARMACEUTICALS INC. (CA) 1997-11-20 WO claimed
US-5770742-A SEROTONIN RECEPTOR SELECTIVITY, MIGRAINES ALLELIX BIOPHARMACEUTICALS INC. (CA) 1998-06-23 US disclosed
WO-1997043281-A1 THIOPHENE- AND FURAN-TRYPTAMINE DERIVATIVES ALLELIX BIOPHARMACEUTICALS INC. (CA) 1997-11-20 WO disclosed