SCHEMBL8784381

SCHEMBL8784381

CC(C)(C)OC(NC=O)(C(=O)O)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
KMT2A Q03164 3/20 0.37
MAPT P10636 1/20 0.37
CYP2C19 P33261 1/20 0.36
HIF1A Q16665 1/20 0.36
GAA P10253 2/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6437393 0.83 KCNN4 (0.46) KCNN4HDAC3HDAC4HDAC1HDAC7
SCHEMBL265970 0.80 MEN1 (0.41) KMT2AGAAMEN1NPC1RAB9A
SCHEMBL6439696 0.79 CYP1A2 (0.40) KCNN4HDAC3HDAC4HDAC1HDAC7
SCHEMBL6435352 0.79 KCNN4 (0.39) KCNN4HDAC3HDAC4HDAC1HDAC7
SCHEMBL6437211 0.76 ALDH1A1 (0.37) KCNN4KMT2AMAPTMEN1ALDH1A1
SCHEMBL4114605 0.75 ALDH1A1 (0.38) KMT2ACYP2C19MEN1NPC1RAB9A
SCHEMBL1455027 0.74 HDAC3 (0.44) KCNN4HDAC3HDAC4HDAC1HDAC7
SCHEMBL1455028 0.74 HDAC3 (0.44) KCNN4HDAC3HDAC4HDAC1HDAC7
SCHEMBL1455851 0.74 HDAC3 (0.44) KCNN4HDAC3HDAC4HDAC1HDAC7
SCHEMBL3786557 0.74 CYP2C19 (0.47) KCNN4HDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0758328-A1 ANTI-CANCER COMPOUNDS CONTAINING CYCLOPENTAQUINAZOLINE RING BTG INTERNATIONAL LIMITED (GB) 1997-02-19 EP disclosed
WO-1995030673-A1 ANTI-CANCER COMPOUNDS CONTAINING CYCLOPENTAQUINAZOLINE RING BRITISH TECHNOLOGY GROUP LIMITED (GB) 1995-11-16 WO disclosed