SCHEMBL878469

SCHEMBL878469

O=C(O)Oc1ccc2c(c1)[C@H](NC(=O)c1ccccc1Cl)CC2

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.58
TAS1R3 Q7RTX0 8/20 0.56
TAS1R1 Q7RTX1 8/20 0.56
TAS1R2 Q8TE23 7/20 0.56
ACHE P22303 9/20 0.46
PDE10A Q9Y233 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL875980 1.00 ALDH1A1 (0.58) ALDH1A1TAS1R3TAS1R1TAS1R2ACHE
SCHEMBL876258 0.89 ALDH1A1 (0.56) ALDH1A1TAS1R3TAS1R1TAS1R2ACHE
SCHEMBL878339 0.89 ALDH1A1 (0.56) ALDH1A1TAS1R3TAS1R1TAS1R2ACHE
SCHEMBL875578 0.84 ACHE (0.46) TAS1R3TAS1R1TAS1R2ACHEPDE10A
SCHEMBL785249 0.83 ALDH1A1 (0.61) ALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL485126 0.83 ALDH1A1 (0.61) ALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL484760 0.83 ALDH1A1 (0.61) ALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL6361268 0.81 ALDH1A1 (0.85) ALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL784965 0.80 ALDH1A1 (0.58) ALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL484334 0.80 ALDH1A1 (0.58) ALDH1A1TAS1R3TAS1R1TAS1R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP disclosed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO disclosed