SCHEMBL8787296

SCHEMBL8787296

CCOC(=O)C1C(=O)N(C)c2cc(OC)c(OC)cc2C1c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
TSHR P16473 3/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
MDM2 Q00987 1/20 0.41
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA9 Q16790 2/20 0.40
HSD17B10 Q99714 1/20 0.40
MAPK1 P28482 3/20 0.40
SIRT3 Q9NTG7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8835165 0.84 TSHR (0.47) ALDH1A1SMN1; SMN2TSHRMEN1CYP1A2
SCHEMBL8784877 0.83 MEN1 (0.44) ALDH1A1SMN1; SMN2TSHRMEN1CYP1A2
SCHEMBL8784942 0.79 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2TSHRMEN1CYP1A2
SCHEMBL8785928 0.74 L3MBTL1 (0.46) ALDH1A1SMN1; SMN2TSHRCYP2C19GAA
SCHEMBL8786585 0.71 L3MBTL1 (0.46) ALDH1A1SMN1; SMN2PDE4DTSHRCYP2C19
SCHEMBL8785879 0.70 L3MBTL1 (0.49) ALDH1A1SMN1; SMN2PDE4BTSHRMEN1
SCHEMBL19124573 0.70 L3MBTL1 (0.43) ALDH1A1SMN1; SMN2TSHRMEN1CYP1A2
SCHEMBL30746805 0.69 MEN1 (0.41) ALDH1A1SMN1; SMN2TSHRMEN1CYP1A2
SCHEMBL29173727 0.69 MEN1 (0.41) ALDH1A1SMN1; SMN2TSHRMEN1CYP1A2
SCHEMBL8784822 0.69 LPAR1 (0.41) SMN1; SMN2MEN1KMT2AKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0585913-B1 Condensed heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-12-29 EP disclosed
US-5700810-A Condensed heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-12-23 US disclosed
US-5482967-A LOWERING CHOLESTEROL TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-01-09 US disclosed
EP-0585913-A2 Condensed heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-09 EP disclosed