SCHEMBL8787882

SCHEMBL8787882

C=CCOC(=O)c1cc(C)ccc1[N+](=O)[O-]

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.49
MAPT P10636 3/20 0.49
CYP3A4 P08684 2/20 0.49
KDM4E B2RXH2 3/20 0.46
KMT2A Q03164 1/20 0.46
TSHR P16473 2/20 0.45
TDP1 Q9NUW8 1/20 0.44
HSD17B10 Q99714 1/20 0.43
GALR2 O43603 1/20 0.40
MITF O75030 1/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
HSP90AA1 P07900 1/20 0.40
HPGD P15428 1/20 0.40
XBP1 P17861 1/20 0.40
CCR6 P51684 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8787481 0.85 CYP3A4 (0.50) ALDH1A1MAPTCYP3A4KDM4EKMT2A
SCHEMBL148384 0.84 MAPT (0.56) ALDH1A1MAPTCYP3A4KDM4EKMT2A
SCHEMBL8759316 0.84 CYP3A4 (0.49) ALDH1A1MAPTCYP3A4KMT2ATSHR
SCHEMBL8787936 0.84 MAPT (0.55) ALDH1A1MAPTCYP3A4KMT2ATSHR
SCHEMBL8787638 0.84 ALDH1A1 (0.50) ALDH1A1MAPTCYP3A4KDM4EKMT2A
SCHEMBL8787027 0.83 CYP3A4 (0.48) ALDH1A1MAPTCYP3A4KDM4EKMT2A
SCHEMBL17368427 0.82 CYP3A4 (0.50) ALDH1A1MAPTCYP3A4KDM4EKMT2A
SCHEMBL8786775 0.81 HTT (0.48) ALDH1A1MAPTCYP3A4KDM4EKMT2A
SCHEMBL11061923 0.81 CYP3A4 (0.64) ALDH1A1MAPTCYP3A4KDM4EKMT2A
SCHEMBL4288671 0.80 CYP3A4 (0.68) ALDH1A1MAPTCYP3A4KMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0508682-B1 Antibiotic carbapenem derivatives ZENECA LTD (GB) 1997-07-23 EP disclosed
US-5541178-A THIENAMYCINS ZENECA LIMITED (GB) 1996-07-30 US disclosed
CN-1066657-A Antimicrobial compounds ICI PLC (GB) 1992-12-02 CN disclosed
WO-1992017481-A1 ANTIBIOTIC CARBAPENEM DERIVATIVES ZENECA LTD. (GB) 1992-10-15 WO disclosed
EP-0508682-A1 Antibiotic carbapenem derivatives ZENECA LIMITED (GB) 1992-10-14 EP disclosed