SCHEMBL8788802

SCHEMBL8788802

CCc1nc2ccc(N(C)S(=O)(=O)c3ccccc3)cc2n1Cc1ccc(-c2ccccc2C#N)cc1

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PPARG P37231 9/20 0.54
ALOX5AP P20292 1/20 0.41
F2 P00734 1/20 0.41
EDNRA P25101 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8788901 0.94 PPARG (0.65) PPARG
SCHEMBL8789752 0.84 PPARG (0.41) PPARG
SCHEMBL8788798 0.81 PPARG (0.54) PPARGALOX5APEDNRA
SCHEMBL7314693 0.81 PPARG (0.56) PPARG
SCHEMBL8848178 0.80 PPARG (0.50) PPARG
SCHEMBL8905159 0.79 F2 (0.38) PPARGF2
SCHEMBL9097162 0.78 AGTR1 (0.68) PPARG
SCHEMBL8789968 0.78 PPARG (0.49) PPARG
SCHEMBL8789971 0.76 PPARG (0.65) PPARGEDNRA
SCHEMBL8788895 0.75 PPARG (0.64) PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0468470-B1 Benzimidazoles, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1997-04-16 EP disclosed
US-5587393-A ANGIOTENSIN ANTAGONIST USEFUL IN TREATING HYPERTENSION DR. KARL THOMAE GMBH (DE) 1996-12-24 US disclosed
US-5385925-A Benzimidazoles, pharmaceutical compositions containing these compounds and processes for preparing them DR. KARL THOMAE GMBH (DE) 1995-01-31 US disclosed
EP-0468470-A1 Benzimidazoles, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1992-01-29 EP disclosed