SCHEMBL8790107

SCHEMBL8790107

N#CSc1nsnc1-c1cccs1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
ALDH1A1 P00352 7/20 0.39
MEN1 O00255 7/20 0.39
KMT2A Q03164 7/20 0.39
KDM4E B2RXH2 6/20 0.39
MAPT P10636 6/20 0.39
HPGD P15428 5/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
POLB P06746 1/20 0.38
ADORA2A P29274 4/20 0.38
ADORA1 P30542 4/20 0.38
ADORA2B P29275 2/20 0.38
PRNP P04156 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9013876 0.81 MEN1 (0.41) CYP1A2CYP2C19CYP3A4CYP2C9ALDH1A1
SCHEMBL2218274 0.76 RPS6KB2 (0.50) CYP1A2CYP2C19CYP3A4CYP2C9ALDH1A1
SCHEMBL8789362 0.75 ERBB2 (0.40) CYP1A2CYP2C9ALDH1A1MEN1KMT2A
SCHEMBL8792142 0.70 MYC (0.52) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL9392461 0.70 CHRM1 (0.38) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL8788935 0.69 MYC (0.50) CYP1A2ALDH1A1MEN1KMT2ANPC1
SCHEMBL8789881 0.69 MYC (0.50) ALDH1A1HPGDADORA2AADORA1
SCHEMBL8790492 0.69 MYC (0.53) KDM4ENPC1RAB9APOLBADORA1
SCHEMBL7217542 0.68 ADORA2A (0.49) CYP1A2CYP2C19CYP3A4CYP2C9ALDH1A1
SCHEMBL8789920 0.68 ADORA1 (0.44) KDM4ENPC1RAB9ASMN1; SMN2ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799216-A1 SUBSTITUTED THIADIAZOLES, COMPOSITIONS CONTAINING THEM AND THEIR USE AS ANTIMICROBIAL AND MARINE ANTIFOULING AGENTS THE DOW CHEMICAL COMPANY (US) 1997-10-08 EP disclosed
WO-1996019467-A1 SUBSTITUTED THIADIAZOLES, COMPOSITIONS CONTAINING THEM AND THEIR USE AS ANTIMICROBIAL AND MARINE ANTIFOULING AGENTS THE DOW CHEMICAL COMPANY (US) 1996-06-27 WO disclosed
US-5488060-A Substituted thiadiazoles, compositions containing them and their use as antimicrobial and marine antifouling agents THE DOW CHEMICAL COMPANY (US) 1996-01-30 US disclosed