SCHEMBL8788935

SCHEMBL8788935

N#CSc1nsnc1-c1ccc(F)cc1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MYC P01106 8/20 0.50
WDR5 P61964 8/20 0.50
ERBB2 P04626 1/20 0.42
ADORA1 P30542 3/20 0.36
ADORA2A P29274 1/20 0.36
KMT2A Q03164 2/20 0.34
CYP1A2 P05177 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
ADORA2B P29275 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
KDM1A O60341 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8789881 0.83 MYC (0.50) MYCWDR5ERBB2ADORA1ADORA2A
SCHEMBL8789633 0.83 MYC (0.50) MYCWDR5ERBB2KMT2ANPSR1
SCHEMBL8789362 0.83 ERBB2 (0.40) MYCWDR5ERBB2ADORA1ADORA2A
SCHEMBL8790492 0.83 MYC (0.53) MYCWDR5ADORA1NPC1RAB9A
SCHEMBL9013799 0.81 MYC (0.35) MYCWDR5ALDH1A1
SCHEMBL8789358 0.80 MYC (0.39) MYCWDR5ERBB2ADORA1ADORA2A
SCHEMBL8792575 0.77 PTGS2 (0.41) MYCWDR5
SCHEMBL27081216 0.75 RAB9A (0.41) MYCWDR5ERBB2ADORA2AKMT2A
SCHEMBL8789377 0.73 IDO1 (0.42) ADORA1ADORA2ACYP1A2ALDH1A1LMNA
SCHEMBL8789920 0.72 ADORA1 (0.44) MYCWDR5ADORA1ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799216-A1 SUBSTITUTED THIADIAZOLES, COMPOSITIONS CONTAINING THEM AND THEIR USE AS ANTIMICROBIAL AND MARINE ANTIFOULING AGENTS THE DOW CHEMICAL COMPANY (US) 1997-10-08 EP disclosed
WO-1996019467-A1 SUBSTITUTED THIADIAZOLES, COMPOSITIONS CONTAINING THEM AND THEIR USE AS ANTIMICROBIAL AND MARINE ANTIFOULING AGENTS THE DOW CHEMICAL COMPANY (US) 1996-06-27 WO disclosed
US-5488060-A Substituted thiadiazoles, compositions containing them and their use as antimicrobial and marine antifouling agents THE DOW CHEMICAL COMPANY (US) 1996-01-30 US disclosed