SCHEMBL879259

SCHEMBL879259

O=C(c1cc(F)cc(C(F)(F)F)c1)c1ccc(I)cn1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 7/20 0.52
KMT2A Q03164 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
CNR2 P34972 1/20 0.38
MAPK1 P28482 1/20 0.38
CES2 O00748 1/20 0.37
GPR52 Q9Y2T5 2/20 0.36
GPBAR1 Q8TDU6 1/20 0.36
PIK3CA P42336 1/20 0.36
LTC4S Q16873 2/20 0.36
CSF1R P07333 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL690788 0.87 VNN1 (0.55) VNN1KMT2AHDAC3HDAC1HDAC2
SCHEMBL842061 0.84 VNN1 (0.49) VNN1LTC4S
SCHEMBL27757817 0.75 CES2 (0.56) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL24851858 0.72 VNN1 (0.46) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL758527 0.71 VNN1 (0.59) VNN1CNR2CES2
SCHEMBL1182880 0.71 VNN1 (0.51) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL1183537 0.69 VNN1 (0.47) VNN1HDAC3HDAC1HDAC2HDAC6
SCHEMBL18286288 0.69 VNN1 (1.00) VNN1
SCHEMBL20185799 0.68 VNN1 (1.00) VNN1
SCHEMBL842548 0.68 CETP (0.41) VNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951690-B1 HETEROCYCLIC CETP INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2012-03-28 EP disclosed