SCHEMBL8792772

SCHEMBL8792772

COc1cc2cc[nH]c2cc1CCC1CCCN1C

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.47
HTR2A P28223 1/20 0.47
HTR1B P28222 3/20 0.44
HTR1A P08908 2/20 0.44
CHRNB4 P30926 4/20 0.43
CHRNA3 P32297 4/20 0.43
BRD4 O60885 1/20 0.40
HTR7 P34969 1/20 0.39
HTR1D P28221 1/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
NPBWR1 P48145 1/20 0.39
MCHR1 Q99705 1/20 0.39
EHMT2 Q96KQ7 1/20 0.39
CHEK1 O14757 1/20 0.39
HTR6 P50406 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22510178 0.76 HRH3 (0.55) HTR1BHTR1ACHRNB4CHRNA3POLB
SCHEMBL8793039 0.74 CHRNB4 (0.49) SLC6A4HTR2ACHRNB4CHRNA3EHMT2
SCHEMBL18475349 0.73 TLR8 (0.51) HTR2APOLB
SCHEMBL8795585 0.72 SLC6A4 (0.42) SLC6A4HTR2AHTR1BHTR1ACHRNB4
SCHEMBL8794935 0.72 CHRNB4 (0.49) CHRNB4CHRNA3
SCHEMBL6740739 0.71 HTR1B (0.51) HTR2AHTR1BHTR1AHTR7HTR1D
SCHEMBL27440375 0.71 TLR8 (0.46) HTR2APOLB
SCHEMBL8705051 0.68 CHRNB4 (0.60) HTR2ACHRNB4CHRNA3
SCHEMBL11455709 0.68 CHRNB4 (0.76) HTR2ACHRNB4CHRNA3EHMT2
SCHEMBL11458219 0.68 CHRNB4 (0.56) CHRNB4CHRNA3EHMT2CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0770079-A1 HETEROBICYCLIC DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-05-02 EP disclosed
EP-0758330-A1 BIPHENYLCARBOXAMIDES USEFUL AS 5-HT1D ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1997-02-19 EP disclosed
WO-1995030675-A1 BIPHENYLCARBOXAMIDES USEFUL AS 5-HT1D ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-11-16 WO disclosed