SCHEMBL8795585

SCHEMBL8795585

COc1cc2c(cc1CCC1CCCN1C)NCC2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.42
CHRNB4 P30926 5/20 0.41
CHRNA3 P32297 5/20 0.41
HTR2A P28223 2/20 0.39
HTR7 P34969 1/20 0.39
CHEK1 O14757 2/20 0.39
UHRF1 Q96T88 1/20 0.38
ACHE P22303 1/20 0.38
HTR1A P08908 2/20 0.37
HTR1B P28222 2/20 0.37
EHMT2 Q96KQ7 1/20 0.37
DRD1 P21728 1/20 0.36
HRH2 P25021 1/20 0.36
HTR2C P28335 1/20 0.36
OPRK1 P41145 1/20 0.36
HTR2B P41595 1/20 0.36
KCNH2 Q12809 1/20 0.36
KCNN2 Q9H2S1 2/20 0.36
KCNN3 Q9UGI6 2/20 0.36
KCNN1 Q92952 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8616789 0.81 SLC6A4 (0.43) SLC6A4HTR2AHTR7DRD1HRH2
SCHEMBL8614215 0.74 HTR7 (0.44) SLC6A4HTR2AHTR7ACHE
SCHEMBL8617442 0.72 CHRNB4 (0.46) CHRNB4CHRNA3
SCHEMBL8792772 0.72 SLC6A4 (0.47) SLC6A4CHRNB4CHRNA3HTR2AHTR7
SCHEMBL8792100 0.72 CHRNB4 (0.46) CHRNB4CHRNA3
SCHEMBL8793039 0.72 CHRNB4 (0.49) SLC6A4CHRNB4CHRNA3HTR2AEHMT2
SCHEMBL8389362 0.70 HTR2A (0.41) SLC6A4HTR2AACHEHTR1BEHMT2
SCHEMBL5564105 0.69 MAOA (0.49) SLC6A4HTR2AHTR2CHTR2B
SCHEMBL3953903 0.66 HTR2A (0.40) HTR2AACHEHTR1AEHMT2HTR2C
SCHEMBL8393003 0.66 NOS1 (0.40) SLC6A4HTR2AACHEHTR1BEHMT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0758330-A1 BIPHENYLCARBOXAMIDES USEFUL AS 5-HT1D ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1997-02-19 EP disclosed
WO-1995030675-A1 BIPHENYLCARBOXAMIDES USEFUL AS 5-HT1D ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-11-16 WO disclosed