SCHEMBL8793473

SCHEMBL8793473

O=c1[nH]c2ccccc2c(=O)n1CCCSc1ccncc1

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.59
HPGD P15428 4/20 0.59
KDM4E B2RXH2 3/20 0.55
MAPK1 P28482 2/20 0.55
HSD17B10 Q99714 2/20 0.55
MPO P05164 2/20 0.54
QPCT Q16769 2/20 0.54
CYP1A2 P05177 1/20 0.50
SMN1; SMN2 Q16637 3/20 0.49
TSHR P16473 2/20 0.47
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.47
HTT P42858 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
GLA P06280 1/20 0.47
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8794286 0.96 ALDH1A1 (0.57) ALDH1A1HPGDKDM4EMAPK1HSD17B10
SCHEMBL8614885 0.81 MAPK1 (0.47) ALDH1A1HPGDMAPK1HSD17B10SMN1; SMN2
Hydrochloric Acid SCHEMBL8619108 0.80 MAPK1 (0.46) ALDH1A1HPGDMAPK1HSD17B10SMN1; SMN2
SCHEMBL8795336 0.79 ALDH1A1 (0.56) ALDH1A1HPGDKDM4EMAPK1HSD17B10
SCHEMBL8616729 0.78 CYP1A2 (0.37) ALDH1A1HPGDKDM4EQPCTCYP1A2
SCHEMBL30159317 0.78 SMN1; SMN2 (0.63) ALDH1A1HPGDKDM4EMAPK1HSD17B10
SCHEMBL8793396 0.78 BACE1 (0.47) CYP1A2MAPTKMT2A
Hydrochloric Acid SCHEMBL8619504 0.78 CYP1A2 (0.36) ALDH1A1HPGDKDM4EQPCTCYP1A2
SCHEMBL8614516 0.77 MAPK1 (0.43) ALDH1A1HPGDMAPK1HSD17B10SMN1; SMN2
Hydrochloric Acid SCHEMBL8794370 0.77 BACE1 (0.46) CYP1A2MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612729-B1 Pyridine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-04-23 EP disclosed
US-5561147-A ANTIINFLAMMATORY AGENT, ANTIPYRETIC, ANALGESICS, ANTIALLERGENS, IMMUNOSUPPRESSANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-10-01 US disclosed
US-5457106-A Antiinflammatory agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-10-10 US disclosed
US-5389658-A Administering as antipyretic, antiinflammatory, analgesic, antiallergic, or immunosupressive agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-02-14 US disclosed
EP-0612729-A2 Pyridine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1994-08-31 EP disclosed
US-5246948-A Antiinflammatory, antipyretic, analgesic, antiallergic, immunosupressing or immunomodulating activity TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-21 US disclosed
EP-0522606-A2 Pyridine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-01-13 EP disclosed