SCHEMBL8795133

SCHEMBL8795133

O=C(O)CCCN1CCC(c2noc3cc(F)ccc23)CC1

nearest known ligand 0.71

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.71
DRD2 P14416 10/20 0.69
SLC6A4 P31645 1/20 0.69
HTR2A P28223 9/20 0.65
HTR1A P08908 2/20 0.65
KCNH2 Q12809 2/20 0.64
HTR2C P28335 1/20 0.64
ADRA1A P35348 1/20 0.64
HRH1 P35367 1/20 0.64
DRD3 P35462 1/20 0.64
HTR6 P50406 1/20 0.64
HTR7 P34969 2/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1545753 0.94 ACHE (0.73) ACHEDRD2SLC6A4HTR2AKCNH2
SCHEMBL7356978 0.92 ACHE (0.71) ACHEDRD2SLC6A4HTR2AHTR1A
SCHEMBL11238900 0.89 DRD2 (0.71) ACHEDRD2SLC6A4HTR2AHTR1A
Fumaric Acid SCHEMBL1545382 0.88 ACHE (0.63) ACHEDRD2SLC6A4HTR2AHTR1A
Hydrochloric Acid SCHEMBL10895287 0.88 DRD2 (0.70) ACHEDRD2SLC6A4HTR2AHTR1A
Ethylene SCHEMBL10894091 0.87 DRD2 (0.69) ACHEDRD2SLC6A4HTR2AHTR1A
SCHEMBL1544799 0.87 ACHE (0.77) ACHEDRD2SLC6A4HTR2AKCNH2
SCHEMBL1545611 0.86 ACHE (0.93) ACHEDRD2SLC6A4HTR2AHTR1A
Fumaric Acid SCHEMBL1545314 0.86 ACHE (0.76) ACHEDRD2SLC6A4HTR2AKCNH2
Fumaric Acid SCHEMBL1545316 0.86 ACHE (0.76) ACHEDRD2SLC6A4HTR2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0730452-A4 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST ROUSSEL PHARMA (US) 1997-03-19 EP disclosed
EP-0730452-A1 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST MARION ROUSSEL, Inc. (US) 1996-09-11 EP disclosed