SCHEMBL8795160

SCHEMBL8795160

COc1cncc(C2=CC(C)(C)Oc3ccc(SC(F)(F)F)cc32)c1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 7/20 0.37
CYP11B2 P19099 7/20 0.37
SLC22A12 Q96S37 1/20 0.34
CYP3A4 P08684 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
BACE1 P56817 4/20 0.33
KCNH2 Q12809 2/20 0.33
CYP17A1 P05093 2/20 0.32
MKNK1 Q9BUB5 1/20 0.31
MKNK2 Q9HBH9 1/20 0.31
RARA P10276 2/20 0.31
RARB P10826 2/20 0.31
RARG P13631 2/20 0.31
CYP1A1 P04798 1/20 0.30
CYP1B1 Q16678 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8794632 0.82 BACE1 (0.35) CYP11B1CYP11B2SLC22A12CYP3A4CYP1A2
SCHEMBL8795368 0.81 RARA (0.33) SLC22A12MKNK1MKNK2RARARARB
SCHEMBL8794705 0.81 RARA (0.35) RARARARBRARG
SCHEMBL8796144 0.79 CYP1A2 (0.34) SLC22A12CYP1A2CYP17A1
SCHEMBL8794799 0.77 SMN1; SMN2 (0.30) RARARARBRARG
SCHEMBL8795475 0.75 SMN1; SMN2 (0.33)
SCHEMBL8795130 0.75 ABL1 (0.32)
SCHEMBL8794583 0.74 SMN1; SMN2 (0.30)
SCHEMBL9378940 0.74 SMN1; SMN2 (0.30)
SCHEMBL8795691 0.73 SMN1; SMN2 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0586405-B1 NOVEL 2H-BENZO[b]PYRANE DERIVATIVES SUBSTITUTED IN THE 4 POSITION BY ARYL OR N-HETEROARYL, PROCESS FOR PRODUCING THEM AND PREPARATIONS CONTAINING THE COMPOUNDS BEIERSDORF LILLY GMBH (DE) 1997-09-10 EP disclosed
EP-0586405-A1 NOVEL 2H-BENZO b]PYRANE DERIVATIVES SUBSTITUTED IN THE 4 POSITION BY ARYL OR N-HETEROARYL, PROCESS FOR PRODUCING THEM AND PREPARATIONS CONTAINING THE COMPOUNDS. BEIERSDORF LILLY GMBH (DE) 1994-03-16 EP disclosed
WO-1992020671-A1 NOVEL 2H-BENZO[b]PYRANE DERIVATIVES SUBSTITUTED IN THE 4 POSITION BY ARYL OR N-HETEROARYL, PROCESS FOR PRODUCING THEM AND PREPARATIONS CONTAINING THE COMPOUNDS BEIERSDORF-LILLY GMBH (DE) 1992-11-26 WO disclosed