SCHEMBL8796387

SCHEMBL8796387

N#Cc1ccccc1OCCCN1CCOCC1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.64
CYP2D6 P10635 2/20 0.57
CYP1A2 P05177 2/20 0.57
CYP2C19 P33261 1/20 0.57
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57
HRH3 Q9Y5N1 2/20 0.56
HRH2 P25021 1/20 0.56
HRH1 P35367 1/20 0.56
TSHR P16473 1/20 0.56
USP2 O75604 1/20 0.55
ALDH1A1 P00352 3/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
DRD1 P21728 1/20 0.50
DRD4 P21917 1/20 0.50
DRD5 P21918 1/20 0.50
CHRM2 P08172 1/20 0.50
CHRM1 P11229 1/20 0.50
HTR2A P28223 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29531493 1.00 KDM4E (0.64) KDM4ECYP2D6CYP1A2CYP2C19MEN1
SCHEMBL8642141 0.93 DRD1 (0.58) KDM4EMEN1KMT2ATSHRALDH1A1
SCHEMBL27885978 0.87 KDM4E (0.55) KDM4ECYP2D6CYP1A2CYP2C19MEN1
SCHEMBL3583983 0.86 CYP2D6 (0.60) KDM4ECYP2D6CYP1A2CYP2C19MEN1
SCHEMBL30303084 0.82 CYP2D6 (0.63) KDM4ECYP2D6CYP1A2CYP2C19MEN1
SCHEMBL27608201 0.82 CYP2D6 (0.63) KDM4ECYP2D6CYP1A2CYP2C19MEN1
SCHEMBL6431609 0.82 HRH3 (0.52) KDM4ECYP2D6CYP1A2CYP2C19MEN1
SCHEMBL6052299 0.82 HRH3 (0.52) KDM4ECYP2D6CYP1A2CYP2C19MEN1
SCHEMBL11162539 0.81 MEN1 (0.64) KDM4ECYP2D6CYP2C19MEN1KMT2A
SCHEMBL11234384 0.79 MEN1 (0.71) KDM4EMEN1KMT2AHRH3HRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5698560-A TREATMENT OF CARDIOVASCULAR DISORDERS; ANTICOAGULANTS; CARDIOTONIC AGENTS; HYPOTENSIVE AGENTS; ARTERIOSCLEROSIS; CYCLIC GMP-SPECIFIC PHOSPHODIESTERASE INHIBITORS KYOWA HAKKO KOGYO CO., LTD. (JP) 1997-12-16 US disclosed
EP-0758653-A1 IMIDAZOQUINAZOLINE DERIVATIVES KYOWA HAKKO KOGYO CO., LTD. (JP) 1997-02-19 EP disclosed