SCHEMBL8797481

SCHEMBL8797481

Cc1ccc2c(c1)C(C(=O)Nc1c(C(C)C)cccc1C(C)C)c1ccccc1CC2

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LPAR1 Q92633 10/20 0.47
LMNA P02545 1/20 0.46
KMT2A Q03164 1/20 0.46
NLRP3 Q96P20 2/20 0.43
TP53 P04637 1/20 0.43
CYP3A4 P08684 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8800082 0.90 KMT2A (0.55) LPAR1LMNAKMT2ASMN1; SMN2
SCHEMBL8797272 0.84 TP53 (0.45) LPAR1LMNAKMT2ANLRP3TP53
SCHEMBL8797711 0.83 LPAR1 (0.49) LPAR1LMNAKMT2ATP53SMN1; SMN2
SCHEMBL8797184 0.83 LPAR1 (0.46) LPAR1LMNAKMT2ANLRP3CYP3A4
SCHEMBL8797886 0.78 LPAR1 (0.42) LPAR1LMNAKMT2ANLRP3TP53
SCHEMBL8797371 0.76 TP53 (0.42) LPAR1LMNAKMT2ANLRP3TP53
SCHEMBL8797526 0.76 TSHR (0.42) LMNAKMT2A
SCHEMBL8797783 0.76 TP53 (0.40) LPAR1KMT2ANLRP3TP53CYP3A4
SCHEMBL8797529 0.76 TP53 (0.46) LPAR1LMNAKMT2ANLRP3TP53
SCHEMBL8798008 0.76 LPAR1 (0.46) LPAR1LMNANLRP3TP53CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0497201-B1 Tricyclic compounds and intermediates thereof KYOWA HAKKO KOGYO KK (JP) 1997-01-15 EP claimed
US-5478835-A Acyl coenzyme A: acyltransferase inhibitors; treatment of hyperlipemia and arteriosclerosis KYOWA HAKKO KOGYO CO., LTD. (JP) 1995-12-26 US claimed
EP-0497201-A1 Tricyclic compounds and intermediates thereof KYOWA HAKKO KOGYO CO., LTD. (JP) 1992-08-05 EP claimed
EP-0497201-B1 Tricyclic compounds and intermediates thereof KYOWA HAKKO KOGYO KK (JP) 1997-01-15 EP disclosed
US-5478835-A Acyl coenzyme A: acyltransferase inhibitors; treatment of hyperlipemia and arteriosclerosis KYOWA HAKKO KOGYO CO., LTD. (JP) 1995-12-26 US disclosed
US-5340807-A Tricyclic compounds and intermediates thereof KYOWA HAKKO KOGYO CO., LTD. (JP) 1994-08-23 US disclosed
EP-0497201-A1 Tricyclic compounds and intermediates thereof KYOWA HAKKO KOGYO CO., LTD. (JP) 1992-08-05 EP disclosed