SCHEMBL8798117

SCHEMBL8798117

O=c1[nH]c(=O)n([C@H]2C[C@@H](CO)[C@@H]2CO)cc1/C=C/Br

nearest known ligand 0.67

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TK1 P04183 6/20 0.67
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
TSHR P16473 1/20 0.58
BLM P54132 1/20 0.58
PMP22 Q01453 1/20 0.58
NPSR1 Q6W5P4 1/20 0.58
TK2 O00142 8/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8689486 1.00 TK1 (0.67) TK1CYP1A2CYP3A4TSHRBLM
SCHEMBL9481617 1.00 TK1 (0.67) TK1CYP1A2CYP3A4TSHRBLM
SCHEMBL9309692 0.91 TK1 (0.76) TK1CYP1A2CYP3A4TSHRBLM
SCHEMBL9309162 0.89 TK1 (0.63) TK1CYP1A2CYP3A4TSHRBLM
SCHEMBL9308662 0.86 TK1 (0.88) TK1CYP1A2CYP3A4TSHRBLM
SCHEMBL8797445 0.85 TK1 (0.50) TK1CYP1A2CYP3A4TSHRBLM
SCHEMBL9734488 0.85 TK1 (0.50) TK1CYP1A2CYP3A4TSHRBLM
SCHEMBL9706093 0.85 TK1 (0.61) TK1CYP1A2CYP3A4TSHRBLM
SCHEMBL10828519 0.83 TK1 (0.65) TK1CYP1A2CYP3A4TSHRBLM
SCHEMBL10827724 0.83 TK1 (0.65) TK1CYP1A2CYP3A4TSHRBLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0335355-B1 Bis-(hydroxymethyl) cyclobutyl purines and pyrimidines SQUIBB & SONS INC (US) 1997-10-01 EP claimed
US-H1142-H Antiviral agent against herpes and varicella-zoster viruses E. R. SQUIBB & SONS, INC. 1993-02-02 US claimed
EP-0484843-A1 An optically active cyclobutyl pyrimidine E.R. SQUIBB & SONS, INC. (US) 1992-05-13 EP claimed
JP-4300872-A None JP disclosed
US-H1142-H Antiviral agent against herpes and varicella-zoster viruses E. R. SQUIBB & SONS, INC. 1993-02-02 US disclosed
US-H1142-H Antiviral agent against herpes and varicella-zoster viruses E. R. SQUIBB & SONS, INC. 1993-02-02 US disclosed
JP-H04300872-A OPTICALLY ACTIVE CYCLOROBUTYL PYRIMIDINE E R SQUIBB & SONS INC 1992-10-23 JP disclosed
US-5130462-A Intermediates for viricides E. R. SQUIBB & SONS, INC. (US) 1992-07-14 US disclosed
US-5126345-A Viricides E. R. SQUIBB & SONS, INC. (US) 1992-06-30 US disclosed
EP-0484843-A1 An optically active cyclobutyl pyrimidine E.R. SQUIBB & SONS, INC. (US) 1992-05-13 EP disclosed
EP-0484843-A1 An optically active cyclobutyl pyrimidine E.R. SQUIBB & SONS, INC. (US) 1992-05-13 EP disclosed