SCHEMBL8798286

SCHEMBL8798286

CO[C@H]1CC[C@H](Nc2cc(Nc3cccc(Cl)c3)ncn2)CC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 8/20 0.59
ERBB3 P21860 3/20 0.59
PIM1 P11309 3/20 0.50
TNNI3K Q59H18 2/20 0.49
PIM2 Q9P1W9 1/20 0.47
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
TUBB4A P04350 1/20 0.43
TUBB P07437 1/20 0.43
TUBA3C P0DPH7 1/20 0.43
TUBA1B P68363 1/20 0.43
TUBA4A P68366 1/20 0.43
TUBB4B P68371 1/20 0.43
TUBB3 Q13509 1/20 0.43
TUBB2A Q13885 1/20 0.43
TUBB8 Q3ZCM7 1/20 0.43
TUBA3E Q6PEY2 1/20 0.43
TUBA1A Q71U36 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8801487 0.87 EGFR (0.50) EGFRERBB3PIM1TNNI3KMEN1
SCHEMBL8799293 0.85 KMO (0.46) EGFRERBB3PIM1MEN1KMT2A
SCHEMBL8799037 0.84 KCNH2 (0.52) EGFRMAPK8MAPK10PDGFRBFBP1
SCHEMBL8799034 0.84 KCNH2 (0.52) EGFRMAPK8MAPK10PDGFRBFBP1
SCHEMBL12481653 0.84 MEN1 (0.57) EGFRERBB3TNNI3KMEN1KMT2A
SCHEMBL8799789 0.82 EGFR (0.52) EGFRERBB3TNNI3KMEN1KMT2A
SCHEMBL8797830 0.82 PRCP (0.60) EGFRERBB3PIM1TNNI3KPRCP
SCHEMBL8798474 0.82 PRCP (0.60) EGFRERBB3PIM1TNNI3KPRCP
SCHEMBL7851792 0.80 EGFR (0.60) EGFRERBB3TNNI3KTUBB4ATUBB
SCHEMBL27345375 0.79 MEN1 (0.69) EGFRERBB3TNNI3KMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed