SCHEMBL8798474

SCHEMBL8798474

CS(=O)(=O)NC1CCC(Nc2cc(Nc3cccc(Cl)c3)ncn2)CC1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRCP P42785 1/20 0.60
TNNI3K Q59H18 9/20 0.56
EGFR P00533 8/20 0.52
PIM1 P11309 2/20 0.52
ERBB3 P21860 2/20 0.51
KCNH2 Q12809 1/20 0.42
S1PR1 P21453 1/20 0.42
CDC7 O00311 1/20 0.42
DAPK3 O43293 1/20 0.42
ROCK2 O75116 1/20 0.42
PRKD3 O94806 1/20 0.42
MAP4K4 O95819 1/20 0.42
PAK4 O96013 1/20 0.42
PRKACA P17612 1/20 0.42
CDK2 P24941 1/20 0.42
FLT3 P36888 1/20 0.42
CDK8 P49336 1/20 0.42
CLK2 P49760 1/20 0.42
GSK3B P49841 1/20 0.42
CDK9 P50750 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8797830 1.00 PRCP (0.60) PRCPTNNI3KEGFRPIM1ERBB3
SCHEMBL8798582 0.88 TNNI3K (0.55) PRCPTNNI3KEGFRPIM1S1PR1
SCHEMBL8798586 0.88 TNNI3K (0.55) PRCPTNNI3KEGFRPIM1S1PR1
SCHEMBL8799768 0.87 TNNI3K (0.56) PRCPTNNI3KEGFRPIM1ERBB3
SCHEMBL8799771 0.87 TNNI3K (0.56) PRCPTNNI3KEGFRPIM1ERBB3
SCHEMBL8801574 0.84 PRCP (0.49) PRCPTNNI3KEGFRPIM1S1PR1
SCHEMBL8799789 0.82 EGFR (0.52) PRCPTNNI3KEGFRERBB3STK3
SCHEMBL12481653 0.82 MEN1 (0.57) TNNI3KEGFRERBB3S1PR1PRKDC
SCHEMBL8798286 0.82 EGFR (0.59) PRCPTNNI3KEGFRPIM1ERBB3
SCHEMBL8319701 0.77 EGFR (0.56) EGFRPIM1MAP4K4CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed