SCHEMBL8798586

SCHEMBL8798586

Cc1cccc(Nc2cc(NC3CCC(NS(C)(=O)=O)CC3)ncn2)c1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TNNI3K Q59H18 14/20 0.55
EGFR P00533 5/20 0.55
PRCP P42785 1/20 0.53
PIM1 P11309 1/20 0.41
USP2 O75604 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C19 P33261 2/20 0.41
CLK4 Q9HAZ1 2/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
S1PR1 P21453 1/20 0.41
LMNA P02545 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8798582 1.00 TNNI3K (0.55) TNNI3KEGFRPRCPPIM1USP2
SCHEMBL8799771 0.88 TNNI3K (0.56) TNNI3KEGFRPRCPPIM1USP2
SCHEMBL8797830 0.88 PRCP (0.60) TNNI3KEGFRPRCPPIM1CLK4
SCHEMBL8798474 0.88 PRCP (0.60) TNNI3KEGFRPRCPPIM1CLK4
SCHEMBL8799768 0.88 TNNI3K (0.56) TNNI3KEGFRPRCPPIM1USP2
SCHEMBL8801574 0.85 PRCP (0.49) TNNI3KEGFRPRCPPIM1USP2
SCHEMBL8798647 0.83 EGFR (0.55) TNNI3KEGFRTSHRMAPK1
SCHEMBL8798643 0.83 EGFR (0.55) TNNI3KEGFRTSHRMAPK1
SCHEMBL8798960 0.82 EGFR (0.54) TNNI3KEGFR
SCHEMBL8798453 0.82 EGFR (0.51) TNNI3KEGFRPIM1CLK4MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed