SCHEMBL8799771

SCHEMBL8799771

CS(=O)(=O)NC1CCC(Nc2cc(Nc3cccc(Br)c3)ncn2)CC1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TNNI3K Q59H18 10/20 0.56
PRCP P42785 1/20 0.52
EGFR P00533 7/20 0.49
ERBB3 P21860 1/20 0.44
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
PIM1 P11309 1/20 0.41
USP2 O75604 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2C19 P33261 2/20 0.40
CLK4 Q9HAZ1 2/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
TSHR P16473 1/20 0.40
S1PR1 P21453 1/20 0.40
LMNA P02545 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8799768 1.00 TNNI3K (0.56) TNNI3KPRCPEGFRERBB3PTGS1
SCHEMBL27330845 0.88 TNNI3K (0.54) TNNI3KEGFRERBB3
SCHEMBL8798586 0.88 TNNI3K (0.55) TNNI3KPRCPEGFRPIM1USP2
SCHEMBL8798582 0.88 TNNI3K (0.55) TNNI3KPRCPEGFRPIM1USP2
SCHEMBL8797830 0.87 PRCP (0.60) TNNI3KPRCPEGFRERBB3PTGS1
SCHEMBL8798474 0.87 PRCP (0.60) TNNI3KPRCPEGFRERBB3PTGS1
SCHEMBL8801574 0.84 PRCP (0.49) TNNI3KPRCPEGFRPIM1USP2
SCHEMBL8801375 0.82 EGFR (0.51) TNNI3KEGFRERBB3
SCHEMBL8801381 0.82 EGFR (0.51) TNNI3KEGFRERBB3
SCHEMBL8800460 0.82 EGFR (0.55) TNNI3KPRCPEGFRERBB3CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed