SCHEMBL8798778

SCHEMBL8798778

COc1ccc2onc(CCNC(C)=O)c(=O)c2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 18/20 0.60
MTNR1B P49286 18/20 0.60
NQO2 P16083 2/20 0.58
HTR2C P28335 2/20 0.53
HTR2B P41595 2/20 0.50
KDM4E B2RXH2 1/20 0.49
MEN1 O00255 1/20 0.49
ALDH1A1 P00352 1/20 0.49
CYP1A1 P04798 1/20 0.49
MPO P05164 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
HTR1A P08908 1/20 0.49
CYP2D6 P10635 1/20 0.49
HPGD P15428 1/20 0.49
RAB9A P51151 1/20 0.49
BLM P54132 1/20 0.49
PMP22 Q01453 1/20 0.49
KMT2A Q03164 1/20 0.49
CYP1B1 Q16678 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9121548 0.92 MTNR1A (0.63) MTNR1AMTNR1BNQO2HTR2CHTR2B
SCHEMBL8798920 0.91 MTNR1A (0.54) MTNR1AMTNR1BNQO2HTR2CHTR2B
SCHEMBL9253876 0.80 MAPT (0.51) HTR2CKDM4EMEN1ALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL9157724 0.79 MAPT (0.50) HTR2CKDM4EMEN1ALDH1A1CYP1A2
SCHEMBL9124933 0.79 MTNR1A (0.65) MTNR1AMTNR1BALDH1A1
SCHEMBL9121405 0.78 MTNR1A (0.56) MTNR1AMTNR1BNQO2
SCHEMBL9119067 0.77 MTNR1A (0.57) MTNR1AMTNR1BNQO2ALDH1A1
SCHEMBL9120386 0.77 MTNR1A (0.67) MTNR1AMTNR1BALDH1A1
SCHEMBL9159270 0.74 MTNR1A (0.65) MTNR1AMTNR1BNQO2HTR2CHTR2B
SCHEMBL9244949 0.74 KDM4E (0.50) KDM4EALDH1A1CYP3A4CYP2D6HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0506539-B1 Heterocyclic alkylamides, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1997-05-02 EP disclosed
US-5436348-A Sleep disorders ADIR ET COMPAGNIE (FR) 1995-07-25 US disclosed
US-5386034-A Treatment of sleeping, psychological and nervous system disorders; anxiolytic agents, ovulation regulators ADIR ET COMPAGNIE (FR) 1995-01-31 US disclosed
US-5322843-A Treating sleep disorders ADIR ET COMPAGNIE (FR) 1994-06-21 US disclosed
EP-0506539-A1 Heterocyclic alkylamides, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1992-09-30 EP disclosed