SCHEMBL8799653

SCHEMBL8799653

FC(F)(F)c1ccc(Nc2cc(NC3CC3)ncn2)cc1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 3/20 0.56
BCR P11274 3/20 0.56
TNNI3K Q59H18 1/20 0.50
TRPV1 Q8NER1 2/20 0.47
MAPK1 P28482 1/20 0.47
EGFR P00533 2/20 0.46
ERBB4 Q15303 1/20 0.46
IRAK4 Q9NWZ3 2/20 0.45
THRB P10828 1/20 0.44
DHODH Q02127 1/20 0.43
MALT1 Q9UDY8 2/20 0.43
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
PIM1 P11309 1/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8799836 0.87 EGFR (0.47) ABL1BCRTNNI3KTRPV1MAPK1
SCHEMBL27317916 0.86 TRPV1 (0.47) ABL1BCRTNNI3KTRPV1EGFR
SCHEMBL27317919 0.84 EGFR (0.49) ABL1BCRMAPK1EGFRMEN1
SCHEMBL8800556 0.81 CDK2 (0.48) TRPV1MAPK1EGFRERBB4IRAK4
SCHEMBL8798532 0.81 KDR (0.46) EGFRERBB4
SCHEMBL27344279 0.81 MEN1 (0.45) MAPK1EGFRIRAK4MEN1KMT2A
SCHEMBL27338340 0.78 KCNQ3 (0.48) ABL1BCRTNNI3KMAPK1EGFR
SCHEMBL29439042 0.77 ABL1 (0.62) ABL1BCRTNNI3KTRPV1EGFR
SCHEMBL27339283 0.77 MEN1 (0.74) TNNI3KEGFRMEN1KMT2A
SCHEMBL27408590 0.77 S1PR1 (0.42) EGFRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed