SCHEMBL27317919

SCHEMBL27317919

Fc1ccc(Nc2cc(NC3CC3)ncn2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.49
ERBB3 P21860 2/20 0.49
MAPK10 P53779 2/20 0.49
CYP1A2 P05177 4/20 0.48
CYP2C19 P33261 4/20 0.48
CYP3A4 P08684 3/20 0.48
CYP2D6 P10635 3/20 0.48
MAPK1 P28482 3/20 0.48
HPGD P15428 1/20 0.48
MEN1 O00255 6/20 0.47
KMT2A Q03164 6/20 0.47
USP2 O75604 2/20 0.47
ALDH1A1 P00352 2/20 0.47
ALOX15 P16050 2/20 0.47
HSD17B10 Q99714 2/20 0.47
CLK4 Q9HAZ1 2/20 0.47
TP53 P04637 1/20 0.47
GLA P06280 1/20 0.47
CYP2C9 P11712 1/20 0.47
LMNA P02545 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27338346 0.86 MEN1 (0.44) EGFRCYP1A2CYP2C19CYP3A4CYP2D6
SCHEMBL27338340 0.85 KCNQ3 (0.48) EGFRERBB3CYP1A2CYP2C19CYP3A4
SCHEMBL27344279 0.84 MEN1 (0.45) EGFRERBB3CYP1A2CYP2C19CYP3A4
SCHEMBL27323499 0.84 MEN1 (0.51) EGFRMAPK10MAPK1MEN1KMT2A
SCHEMBL8799653 0.84 ABL1 (0.56) EGFRMAPK1MEN1KMT2AABL1
SCHEMBL27408590 0.81 S1PR1 (0.42) EGFRERBB3CYP1A2CYP3A4CYP2D6
SCHEMBL27339283 0.81 MEN1 (0.74) EGFRERBB3MEN1KMT2AALDH1A1
SCHEMBL27339284 0.81 GPR119 (0.42) EGFRERBB3CYP1A2CYP2C19CYP3A4
SCHEMBL27317916 0.81 TRPV1 (0.47) EGFRCYP1A2CYP2C19CYP3A4CYP2D6
SCHEMBL8798532 0.79 KDR (0.46) EGFRS1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1047778-C Pyrimido [5-4-d] pyrimidines, drugs containing these compounds, their use and process for preparing them THOMAE GMBH DR K (DE) 1999-12-29 CN disclosed