SCHEMBL8799684

SCHEMBL8799684

COC(=O)CO[C@H]1CC[C@H](Nc2cc(Nc3ccc(F)c(Cl)c3)ncn2)CC1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.47
EGFR P00533 12/20 0.43
MAPKAPK2 P49137 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
MAPT P10636 1/20 0.42
PRCP P42785 1/20 0.42
ERBB2 P04626 2/20 0.40
ALDH1A1 P00352 1/20 0.40
ERBB4 Q15303 1/20 0.40
ROCK2 O75116 1/20 0.40
CDK2 P24941 1/20 0.40
MAPK9 P45984 1/20 0.40
GSK3B P49841 1/20 0.40
MAP2K1 Q02750 1/20 0.40
MAPKAPK5 Q8IW41 1/20 0.40
S1PR1 P21453 1/20 0.39
ERBB3 P21860 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8798668 0.91 KCNH2 (0.46) KCNH2EGFRMAPKAPK2MEN1KMT2A
SCHEMBL8798680 0.91 KCNH2 (0.46) KCNH2EGFRMAPKAPK2MEN1KMT2A
SCHEMBL8799034 0.85 KCNH2 (0.52) KCNH2EGFRMAPKAPK2ERBB2ROCK2
SCHEMBL8799037 0.85 KCNH2 (0.52) KCNH2EGFRMAPKAPK2ERBB2ROCK2
SCHEMBL7858523 0.85 KCNH2 (0.47) KCNH2EGFRMAPKAPK2MEN1KMT2A
SCHEMBL7701772 0.84 KCNH2 (0.49) KCNH2EGFRMAPKAPK2MEN1KMT2A
SCHEMBL7701769 0.84 KCNH2 (0.49) KCNH2EGFRMAPKAPK2MEN1KMT2A
SCHEMBL8318239 0.84 KCNH2 (0.51) KCNH2EGFRMAPKAPK2MEN1KMT2A
SCHEMBL8318242 0.84 KCNH2 (0.51) KCNH2EGFRMAPKAPK2MEN1KMT2A
SCHEMBL7691002 0.83 ERBB2 (0.48) KCNH2EGFRMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed