SCHEMBL8799700

SCHEMBL8799700

CC(=O)N[C@H]1CC[C@H](Nc2cc(Nc3cccc([N+](=O)[O-])c3)ncn2)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.53
TNNI3K Q59H18 1/20 0.53
FLT3 P36888 1/20 0.49
TYRO3 Q06418 1/20 0.49
MERTK Q12866 1/20 0.49
GAS6 Q14393 1/20 0.49
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CCNT1 O60563 2/20 0.46
CDK9 P50750 2/20 0.46
PIK3CA P42336 1/20 0.44
MTOR P42345 1/20 0.44
PRKDC P78527 1/20 0.44
PKM P14618 1/20 0.44
ROCK1 Q13464 1/20 0.43
ABCG2 Q9UNQ0 2/20 0.43
ABCC1 P33527 1/20 0.43
CTSL P07711 2/20 0.43
CTSB P07858 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12485644 0.85 CTSL (0.57) EGFRTNNI3KFLT3TYRO3MERTK
SCHEMBL27322786 0.84 EGFR (0.54) EGFRTNNI3KFLT3TYRO3MERTK
SCHEMBL8798751 0.84 EGFR (0.51) EGFRTNNI3KNPC1RAB9ASMN1; SMN2
SCHEMBL8798748 0.84 EGFR (0.51) EGFRTNNI3KNPC1RAB9ASMN1; SMN2
SCHEMBL27423214 0.83 EGFR (0.55) EGFRTNNI3KFLT3TYRO3MERTK
SCHEMBL27338343 0.83 CTSL (0.58) EGFRTNNI3KFLT3TYRO3MERTK
SCHEMBL8799789 0.83 EGFR (0.52) EGFRTNNI3KNPC1RAB9APRKDC
SCHEMBL8800460 0.83 EGFR (0.55) EGFRTNNI3KIRAK4
SCHEMBL8800238 0.80 EGFR (0.47) EGFRFLT3TYRO3MERTKGAS6
SCHEMBL8315077 0.78 FLT3 (0.47) EGFRFLT3TYRO3MERTKGAS6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed