SCHEMBL8799703

SCHEMBL8799703

CCc1ccc2c(c1)c(-c1ccc3c(c1)OCO3)c(OC(=O)O)c(=O)n2Cc1cc(OC)ccc1OC

nearest known ligand 0.66

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 14/20 0.66
EDNRA P25101 9/20 0.55
KMT2A Q03164 1/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8798624 0.93 EDNRB (0.63) EDNRBEDNRAKMT2AKDM4EALDH1A1
SCHEMBL8578754 0.89 EDNRB (0.83) EDNRBEDNRAKDM4EALDH1A1
SCHEMBL8578633 0.87 EDNRB (0.73) EDNRBEDNRAKMT2A
SCHEMBL8798655 0.85 EDNRB (0.67) EDNRBEDNRAKMT2AKDM4EALDH1A1
SCHEMBL8798670 0.83 EDNRB (0.63) EDNRBEDNRA
SCHEMBL8798379 0.83 EDNRB (0.81) EDNRBEDNRA
SCHEMBL8798982 0.82 EDNRB (0.78) EDNRBEDNRA
SCHEMBL8798255 0.81 EDNRB (0.79) EDNRBEDNRAKDM4EALDH1A1
SCHEMBL8798525 0.81 EDNRB (0.61) EDNRBEDNRA
SCHEMBL8798374 0.80 EDNRB (0.64) EDNRBEDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757039-A1 Endothelin receptor antagonists MERCK PATENT GmbH (DE) 1997-02-05 EP disclosed