SCHEMBL8799995

SCHEMBL8799995

NC1CCN(c2cc(Nc3ccc(F)c(Cl)c3)ncn2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.51
KDR P35968 4/20 0.49
EGFR P00533 3/20 0.48
ERBB2 P04626 2/20 0.48
LCK P06239 1/20 0.48
MAPK1 P28482 1/20 0.47
MALT1 Q9UDY8 3/20 0.46
KCNH2 Q12809 1/20 0.45
CDK2 P24941 4/20 0.45
MAPKAPK2 P49137 4/20 0.45
GALR2 O43603 1/20 0.45
PAK4 O96013 1/20 0.44
PAK1 Q13153 1/20 0.44
ROCK2 O75116 1/20 0.44
MAPK9 P45984 1/20 0.44
GSK3B P49841 1/20 0.44
MAP2K1 Q02750 1/20 0.44
MAPKAPK5 Q8IW41 1/20 0.44
ABL1 P00519 1/20 0.43
BCR P11274 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8799651 0.83 GALR2 (0.45) KDREGFRMAPK1MALT1GALR2
SCHEMBL7854183 0.81 EGFR (0.43) CHEK1EGFRERBB2MAPK1MALT1
SCHEMBL8571074 0.80 GRM1 (0.54) KDREGFRERBB2LCKGRM1
SCHEMBL4350714 0.80 GRM1 (0.62) KDREGFRERBB2LCKGRM1
SCHEMBL7852078 0.80 MALT1 (0.45) EGFRERBB2MALT1MAPT
SCHEMBL8597285 0.80 EGFR (0.52) KDREGFRERBB2LCKKCNH2
SCHEMBL7846724 0.79 KCNH2 (0.66) KDREGFRERBB2LCKMAPK1
SCHEMBL7851279 0.79 KCNH2 (0.66) KDREGFRERBB2LCKMAPK1
SCHEMBL7844610 0.79 LIMK1 (0.46) EGFRMAPK1MALT1GALR2ROCK2
SCHEMBL25385769 0.78 KCNH2 (0.69) KDREGFRERBB2LCKMALT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed