SCHEMBL8799651

SCHEMBL8799651

O=C1CCN(c2cc(Nc3ccc(F)c(Cl)c3)ncn2)CC1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GALR2 O43603 1/20 0.45
MAPK1 P28482 1/20 0.45
ABL1 P00519 1/20 0.43
BCR P11274 1/20 0.43
MALT1 Q9UDY8 2/20 0.42
SCN9A Q15858 2/20 0.41
EGFR P00533 5/20 0.41
KDR P35968 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
AURKA O14965 2/20 0.41
AURKB Q96GD4 2/20 0.41
GRM1 Q13255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KMO O15229 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8799995 0.83 CHEK1 (0.51) GALR2MAPK1ABL1BCRMALT1
SCHEMBL7853244 0.81 HPGD (0.48) GALR2MALT1EGFRAURKAAURKB
SCHEMBL7844610 0.80 LIMK1 (0.46) GALR2MAPK1MALT1SCN9AEGFR
SCHEMBL7853525 0.79 MCHR1 (0.47) EGFRAURKAAURKBKMO
SCHEMBL7854183 0.78 EGFR (0.43) GALR2MAPK1ABL1BCRMALT1
SCHEMBL7852431 0.78 LIMK1 (0.48) GALR2MAPK1ABL1BCRMALT1
SCHEMBL7852078 0.77 MALT1 (0.45) MALT1SCN9AEGFRKMO
SCHEMBL7845264 0.77 EGFR (0.47) GALR2EGFRKDRAURKAAURKB
SCHEMBL27401069 0.76 KMO (0.52) GALR2ABL1BCRALDH1A1RAB9A
SCHEMBL7855449 0.76 EGFR (0.46) GALR2ABL1BCRSCN9AEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed