SCHEMBL8801485

SCHEMBL8801485

CC[C@H](C)[C@H](NC(=O)CC1OC1C(Cc1ccccc1)NC(=O)[C@@H](CC(N)=O)NC(=O)c1ccc2ccccc2n1)C(=O)NCc1nc2ccccc2[nH]1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 6/20 0.68
REN P00797 3/20 0.45
CTSE P14091 1/20 0.45
PSMB5 P28074 2/20 0.39
HDAC1 Q13547 1/20 0.38
CYP3A4 P08684 4/20 0.38
ABCC3 O15438 1/20 0.38
ABCC4 O15439 1/20 0.38
CACNA1F O60840 1/20 0.38
ABCB11 O95342 1/20 0.38
ABCB1 P08183 1/20 0.38
HTR1A P08908 1/20 0.38
DRD2 P14416 1/20 0.38
TACR2 P21452 1/20 0.38
TBXAS1 P24557 1/20 0.38
OPRM1 P35372 1/20 0.38
DRD3 P35462 1/20 0.38
AVPR1A P37288 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8800288 0.94 CTSD (0.73) CTSDRENCTSEHDAC1CYP3A4
SCHEMBL8802750 0.92 CTSD (0.76) CTSDRENCTSEPSMB5HDAC1
SCHEMBL8801937 0.88 CTSD (0.78) CTSDRENCTSEPSMB5HDAC1
SCHEMBL7313674 0.88 CTSD (0.80) CTSDRENCTSEPSMB5HDAC1
SCHEMBL8801445 0.88 CTSD (0.70) CTSDRENCTSEPSMB5HDAC1
SCHEMBL8800743 0.87 CTSD (0.59) CTSDRENPSMB5HDAC1CYP3A4
SCHEMBL8801592 0.86 CTSD (0.77) CTSDRENCTSEPSMB5CYP3A4
SCHEMBL8800871 0.83 CTSD (0.86) CTSDRENCTSEPSMB5HDAC1
SCHEMBL8800938 0.82 CTSD (0.74) CTSDRENCTSEHDAC1CYP3A4
SCHEMBL8801929 0.81 CTSD (0.82) CTSDRENCTSEHDAC1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0601486-B1 Cis-epoxide derivatives useful as irreversible HIV protease inhibitors and process and intermediates for their preparation LUCKY LTD (KR) 1997-10-29 EP claimed
EP-0601486-A1 Cis-epoxide derivatives useful as irreversible HIV protease inhibitors and process and intermediates for their preparation LUCKY LTD. (KR) 1994-06-15 EP claimed