SCHEMBL8801611

SCHEMBL8801611

O=C(O)C=Cc1ccc(/C=C/c2cccnc2)nc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.59
NPC1 O15118 2/20 0.59
MAPT P10636 2/20 0.59
KDM4E B2RXH2 2/20 0.59
JUN P05412 1/20 0.59
NFKB1 P19838 1/20 0.59
MAPK1 P28482 1/20 0.59
GPR55 Q9Y2T6 1/20 0.59
TBXAS1 P24557 3/20 0.58
KMT2A Q03164 2/20 0.54
MEN1 O00255 1/20 0.54
CYP11B1 P15538 1/20 0.53
CYP11B2 P19099 1/20 0.53
P4HTM Q9NXG6 1/20 0.53
PFKFB3 Q16875 1/20 0.52
CYP1A1 P04798 3/20 0.51
CYP1A2 P05177 3/20 0.51
CYP1B1 Q16678 3/20 0.51
PIM2 Q9P1W9 1/20 0.49
CYP3A4 P08684 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6642060 1.00 RAB9A (0.59) RAB9ANPC1MAPTKDM4EJUN
SCHEMBL6642064 1.00 RAB9A (0.59) RAB9ANPC1MAPTKDM4EJUN
SCHEMBL2865108 0.90 CYP11B1 (0.60) RAB9ANPC1MAPTKDM4EJUN
SCHEMBL755249 0.87 RAB9A (0.76) RAB9ANPC1MAPTKDM4EJUN
SCHEMBL334615 0.87 RAB9A (0.76) RAB9ANPC1MAPTKDM4EJUN
SCHEMBL334614 0.87 RAB9A (0.76) RAB9ANPC1MAPTKDM4EJUN
SCHEMBL29416684 0.87 RAB9A (0.76) RAB9ANPC1MAPTKDM4EJUN
Hydrochloric Acid SCHEMBL27850886 0.86 RAB9A (0.73) RAB9ANPC1MAPTKDM4EJUN
SCHEMBL10898888 0.86 RAB9A (0.73) RAB9ANPC1MAPTKDM4EJUN
Hydrochloric Acid SCHEMBL10810828 0.86 RAB9A (0.73) RAB9ANPC1MAPTKDM4EJUN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0807105-A1 PYRIDOPYRIMIDONES, QUINOLINES AND FUSED N-HERETOCYCLES AS BRADYKININ ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-11-19 EP disclosed