SCHEMBL8801694

SCHEMBL8801694

CCc1cc(=O)c2c(NCc3ccccc3)c(F)c(F)c(F)c2n1-c1cc(NC=O)c(F)cc1F

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA7 P43166 1/20 0.32
CA13 Q8N1Q1 1/20 0.32
IKBKB O14920 1/20 0.31
AURKA O14965 1/20 0.31
CHUK O15111 1/20 0.31
MAPK13 O15264 1/20 0.31
DAPK3 O43293 1/20 0.31
PRKCG P05129 1/20 0.31
PIM1 P11309 1/20 0.31
CDK2 P24941 1/20 0.31
MARK3 P27448 1/20 0.31
AKT1 P31749 1/20 0.31
AKT2 P31751 1/20 0.31
MAPKAPK2 P49137 1/20 0.31
GSK3A P49840 1/20 0.31
NEK2 P51955 1/20 0.31
PLK1 P53350 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29950022 0.60 CA2 (0.66) CA12CA1CA2CA7CA13
SCHEMBL28228895 0.59 CA2 (0.56) CA12CA1CA2CA7CA13
SCHEMBL15578977 0.55 MEN1 (0.43) TP53MAPTSMN1; SMN2HDAC1HDAC8
SCHEMBL13720 0.54 KDM5A (0.34) CA12CA1CA2MAPT
SCHEMBL9501324 0.54 TSHR (0.46) CA12CA1CA2CA7CA13
SCHEMBL10546027 0.53 KMT2A (0.50) CA12CA1CA2CA7CA13
SCHEMBL15470920 0.53 CA2 (0.55) CA12CA1CA2CA7CA13
SCHEMBL3747115 0.53 MAPKAPK2 (0.66) CA12CA1CA2CA7CA13
SCHEMBL21371036 0.52 CA2 (0.58) CA12CA1CA2CA7CA13
SCHEMBL22909578 0.52 CA2 (0.61) CA12CA1CA2CA7CA13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0787720-A1 NOVEL PYRIDONECARBOXYLATE DERIVATIVE OR SALT THEREOF AND ANTIBACTERIAL CONTAINING THE SAME AS ACTIVE INGREDIENT WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1997-08-06 EP disclosed