SCHEMBL8802005

SCHEMBL8802005

O=C(CN1CCc2sccc2C1)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.53
KDM4E B2RXH2 2/20 0.53
CASP1 P29466 1/20 0.53
CYP2C19 P33261 2/20 0.51
DRD3 P35462 2/20 0.51
HTR2B P41595 2/20 0.51
USP2 O75604 1/20 0.51
ABCB11 O95342 1/20 0.51
LMNA P02545 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
ADRA2A P08913 1/20 0.51
ADORA3 P0DMS8 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
ADRB3 P13945 1/20 0.51
ADRA2B P18089 1/20 0.51
ADRA2C P18825 1/20 0.51
CYP2B6 P20813 1/20 0.51
DRD1 P21728 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10623034 0.86 DRD3 (0.59) ALDH1A1KDM4ECYP2C19DRD3HTR2B
SCHEMBL6369881 0.84 ALDH1A1 (0.50) ALDH1A1KDM4ECASP1CYP2C19DRD3
SCHEMBL5242060 0.80 ALDH1A1 (0.49) ALDH1A1KDM4ECASP1CYP2C19DRD3
Water SCHEMBL11003040 0.79 ALDH1A1 (0.47) ALDH1A1KDM4ECASP1CYP2C19DRD3
SCHEMBL8801055 0.79 CYP2C19 (0.47) ALDH1A1KDM4ECASP1CYP2C19DRD3
SCHEMBL3381087 0.76 ALDH1A1 (0.55) ALDH1A1KDM4ECASP1CYP2C19DRD3
SCHEMBL28687701 0.76 CYP2C19 (0.55) ALDH1A1KDM4ECASP1CYP2C19DRD3
SCHEMBL6631313 0.76 CYP2C19 (0.49) ALDH1A1KDM4ECASP1CYP2C19DRD3
SCHEMBL3992345 0.75 HSP90AA1 (0.52) ALDH1A1LMNASMN1; SMN2AKR1C3PRMT5
SCHEMBL30546565 0.75 ALDH1A1 (0.57) ALDH1A1KDM4ECASP1CYP2C19DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0522956-B1 Preparation of 2-(2-thienyl) ethylamine and synthesis of thieno [3,2-C] pyridine derivatives therefrom SANOFI SA (FR) 1997-02-05 EP disclosed
US-5191090-A Preparation of 2-(2'-thienyl)ethylamine derivatives and synthesis of thieno[3,2-c]pyridine derivatives therefrom SYNTEX (U.S.A.) INC. (US) 1993-03-02 US disclosed
EP-0522956-A2 Preparation of 2-(2-thienyl) ethylamine and synthesis of thieno [3,2-C] pyridine derivatives therefrom SANOFI (FR) 1993-01-13 EP disclosed
US-5068360-A Preparation of 2-(2'-thienyl)ethylamine derivatives and synthesis of thieno(3,2-C)pyridine derivatives therefrom SYNTEX (U.S.A.) INC. (US) 1991-11-26 US disclosed
EP-0439404-A2 Preparation of 2-(2'-thienyl) alkylamines and derivatives thereof and synthesis of 4,5,6,7- thieno [3,2-c] pyridine derivatives therefrom SANOFI (FR) 1991-07-31 EP disclosed
US-4997945-A Ticlopidine intermediate SYNTEX (U.S.A.) INC. (US) 1991-03-05 US disclosed
US-4906756-A 2-(2-nitrovinyl)thiophene reduction and synthesis of thieno[3,2-c]pyridine derivatives SYNTEX (U.S.A.) INC. (US) 1990-03-06 US disclosed
EP-0342118-A1 2-(2-nitrovinyl)thiophene reduction and synthesis of thieno (3,2-c)pyridine derivatives ELF SANOFI (FR) 1989-11-15 EP disclosed