SCHEMBL8802467

SCHEMBL8802467

COc1ccc2ncc(C(=O)OCC3CCCCN3C)cc2c1

nearest known ligand 0.70

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 10/20 0.70
CHRNA4 P43681 9/20 0.70
CHRNA7 P36544 7/20 0.70
CHRNA5 P30532 3/20 0.51
HPGDS O60760 4/20 0.48
CHRNB4 P30926 2/20 0.47
CHRNA3 P32297 2/20 0.47
CHRNB1 P11230 1/20 0.45
CHRNB3 Q05901 1/20 0.45
ALDH1A1 P00352 1/20 0.43
F2 P00734 1/20 0.43
GLA P06280 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL620719 0.78 ALDH1A1 (0.46) CHRNB2CHRNA4CHRNA7HPGDSALDH1A1
SCHEMBL620720 0.78 ALDH1A1 (0.46) CHRNB2CHRNA4CHRNA7HPGDSALDH1A1
SCHEMBL545163 0.76 MAOB (0.65) HPGDSALDH1A1F2GLAHPGD
SCHEMBL20799517 0.73 ALDH1A1 (0.62) HPGDSALDH1A1F2GLAHPGD
SCHEMBL622650 0.71 HPGDS (0.49) HPGDS
SCHEMBL622649 0.71 HPGDS (0.49) HPGDS
SCHEMBL61795 0.69 ALDH1A1 (0.64) HPGDSALDH1A1F2GLAHPGD
SCHEMBL4407431 0.69 ALDH1A1 (0.68) HPGDSALDH1A1F2GLAHPGD
SCHEMBL1353255 0.69 HPGDS (0.63) HPGDSALDH1A1F2GLAHPGD
SCHEMBL8802477 0.69 HPGDS (0.45) HPGDSALDH1A1F2GLAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0499995-B1 Piperidine derivatives NISSHIN FLOUR MILLING CO (JP) 1997-01-02 EP disclosed
US-5246945-A 5-hydroxytryptamine antagonist for nervous system disorders NISSHIN FLOUR MILLING CO., LTD. (JP) 1993-09-21 US disclosed
EP-0499995-A2 Piperidine derivatives NISSHIN FLOUR MILLING CO., LTD. (JP) 1992-08-26 EP disclosed