SCHEMBL8805345

SCHEMBL8805345

O=C(c1ccc(F)cc1)C1CCN(CCCOc2cc(=O)oc3ccccc23)CC1

nearest known ligand 0.67

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.54
KDM4E B2RXH2 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
HTR2A P28223 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8686164 0.84 HTR2A (0.52) KDM4ECYP1A2CYP3A4CYP2D6HTR2A
SCHEMBL6253491 0.81 HTR2A (0.60) KDM4ECYP1A2CYP3A4CYP2D6HTR2A
SCHEMBL8806438 0.79 KCNH2 (0.62) MAOBHTR2A
SCHEMBL8807400 0.79 HTR2A (0.57) KDM4ECYP1A2CYP3A4CYP2D6HTR2A
SCHEMBL8804878 0.79 DRD2 (0.61) MAOB
SCHEMBL1583103 0.78 KDM4E (0.69) MAOBKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL8805189 0.77 HTR2A (0.55) KDM4ECYP1A2CYP3A4CYP2D6HTR2A
SCHEMBL8805723 0.77 HTR2A (0.65) KDM4ECYP1A2CYP3A4CYP2D6HTR2A
SCHEMBL29794227 0.77 MAOB (0.69) MAOB
SCHEMBL29046355 0.77 MAOB (0.69) MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0751936-A1 NEW 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES USEFUL AS MEDICAMENTS ACTING ON THE GLUTAMATE RECEPTOR SCHERING AKTIENGESELLSCHAFT (DE) 1997-01-08 EP claimed
WO-1995025721-A1 NEW 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES USEFUL AS MEDICAMENTS ACTING ON THE GLUTAMATE RECEPTOR SCHERING AKTIENGESELLSCHAFT (DE) 1995-09-28 WO claimed
EP-0751936-A1 NEW 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES USEFUL AS MEDICAMENTS ACTING ON THE GLUTAMATE RECEPTOR SCHERING AKTIENGESELLSCHAFT (DE) 1997-01-08 EP disclosed
WO-1995025721-A1 NEW 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES USEFUL AS MEDICAMENTS ACTING ON THE GLUTAMATE RECEPTOR SCHERING AKTIENGESELLSCHAFT (DE) 1995-09-28 WO disclosed