SCHEMBL8806399

SCHEMBL8806399

Cc1cc(C)nc(NC(=O)C=Cc2c(Cc3ccccc3)[nH]c3ccccc23)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.51
NPC1 O15118 5/20 0.51
RAB9A P51151 5/20 0.51
MAPT P10636 5/20 0.51
KDM4E B2RXH2 4/20 0.51
MEN1 O00255 4/20 0.51
KMT2A Q03164 4/20 0.51
SMN1; SMN2 Q16637 4/20 0.51
HPGD P15428 5/20 0.45
CYP1A2 P05177 3/20 0.45
CYP2C19 P33261 3/20 0.45
CYP2D6 P10635 2/20 0.45
CASP3 P42574 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
SENP8 Q96LD8 1/20 0.45
SENP7 Q9BQF6 1/20 0.45
SENP6 Q9GZR1 1/20 0.45
TDP1 Q9NUW8 3/20 0.40
CYP3A4 P08684 2/20 0.40
TSHR P16473 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8805183 0.79 CYP3A4 (0.49) ALDH1A1RAB9AMAPTKDM4EMEN1
SCHEMBL8807288 0.78 MEN1 (0.49) ALDH1A1NPC1RAB9AMAPTKDM4E
SCHEMBL8804361 0.75 KMT2A (0.48) ALDH1A1MAPTKDM4EMEN1KMT2A
SCHEMBL8803840 0.74 KMT2A (0.49) ALDH1A1MAPTKDM4EMEN1KMT2A
SCHEMBL8806394 0.72 MAPT (0.60) ALDH1A1NPC1RAB9AMAPTKDM4E
SCHEMBL8805502 0.69 MAPK1 (0.44) ALDH1A1NPC1RAB9AMAPTKDM4E
SCHEMBL10871902 0.69 MAPT (0.48) ALDH1A1NPC1RAB9AMAPTKDM4E
SCHEMBL28863000 0.68 AHR (0.54) ALDH1A1NPC1KDM4EMEN1KMT2A
SCHEMBL8806760 0.68 RAB9A (0.62) ALDH1A1NPC1RAB9AMAPTKDM4E
SCHEMBL8806770 0.68 RAB9A (0.62) ALDH1A1NPC1RAB9AMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775131-A2 INDOL, INDAZOL, PYRIDOPYRROL AND PYRIDOPYRAZOL DERIVATIVES WITH ANTI-ASTHMATIC, ANTI-ALLERGIC, ANTI-INFLAMMATORY AND IMMUNOMODULATING EFFECTS ASTA Medica Aktiengesellschaft (DE) 1997-05-28 EP disclosed
WO-1996004266-A2 INDOL, INDAZOL, PYRIDOPYRROL AND PYRIDOPYRAZOL DERIVATIVES WITH ANTI-ASTHMATIC, ANTI-ALLERGIC, ANTI-INFLAMMATORY AND IMMUNOMODULATING EFFECTS ASTA MEDICA AKTIENGESELLSCHAFT (DE) 1996-02-15 WO disclosed