Bicarbonate

Bicarbonate

SCHEMBL8806909

Cn1c(=O)c(=O)[nH]c2cc([N+](=O)[O-])c3ccccc3c21.O=C(O)O

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.47
PARP1 P09874 9/20 0.44
GRIK1 P39086 3/20 0.42
GRIK2 Q13002 3/20 0.42
GRIK3 Q13003 3/20 0.42
GRIK4 Q16099 3/20 0.42
GRIK5 Q16478 3/20 0.42
GRIA1 P42261 2/20 0.41
GRIA2 P42262 2/20 0.41
GRIA3 P42263 2/20 0.41
GRIA4 P48058 2/20 0.41
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
BLM P54132 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL8807930 0.82 GRIK1 (0.61) PARP1GRIK1GRIK2GRIK3GRIK4
SCHEMBL9396484 0.81 GRIA1 (0.46) SIRT2PARP1GRIK1GRIK2GRIK3
SCHEMBL8621659 0.81 SIRT2 (0.43) SIRT2PARP1GRIK1GRIK2GRIK3
SCHEMBL8618891 0.81 GRIK1 (0.57) SIRT2GRIK1GRIK2GRIK3GRIK4
Bicarbonate SCHEMBL8807164 0.81 SIRT2 (0.47) SIRT2PARP1GRIK1GRIK2GRIK3
SCHEMBL8805561 0.79 SIRT2 (0.41) SIRT2GRIK1GRIK2GRIK3GRIK4
SCHEMBL8621742 0.76 SIRT2 (0.43) SIRT2PARP1GRIK1GRIK2GRIK3
SCHEMBL3691418 0.76 KMT2A (0.65) SIRT2PARP1GRIK1GRIK2GRIK3
SCHEMBL9749640 0.76 MEN1 (0.43) SIRT2GRIK1GRIK2GRIK3GRIK4
SCHEMBL8619770 0.75 GRIA1 (0.44) SIRT2GRIK1GRIK2GRIK3GRIK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696289-B1 BENZO[F]QUINOXALINDIONE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN DRUGS SCHERING AG (DE) 1997-03-12 EP claimed
EP-0696289-B1 BENZO[F]QUINOXALINDIONE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN DRUGS SCHERING AG (DE) 1997-03-12 EP disclosed
WO-1994025470-A1 BENZO[F]QUINOXALINDIONE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN DRUGS SCHERING AKTIENGESELLSCHAFT (DE) 1994-11-10 WO disclosed