SCHEMBL8807285

SCHEMBL8807285

COc1cc2ncnc(Nc3ccc(CS(=O)(=O)c4ccccc4)cc3)c2cc1OC

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 12/20 0.67
KDR P35968 6/20 0.67
RET P07949 2/20 0.67
LCK P06239 3/20 0.66
LRRK2 Q5S007 2/20 0.64
PIK3CD O00329 1/20 0.64
PIK3CA P42336 1/20 0.64
PIK3CB P42338 1/20 0.64
PIK3CG P48736 1/20 0.64
RIPK2 O43353 2/20 0.63
EPHB2 P29323 1/20 0.63
AURKA O14965 1/20 0.60
AURKB Q96GD4 1/20 0.60
SRC P12931 1/20 0.59
FLT1 P17948 1/20 0.58
GAK O14976 1/20 0.58
STK10 O94804 1/20 0.58
FLT3 P36888 1/20 0.58
JAK3 P52333 1/20 0.58
AAK1 Q2M2I8 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8807988 0.96 EGFR (0.67) EGFRKDRRETLCKLRRK2
SCHEMBL8807167 0.86 EGFR (0.75) EGFRKDRRETLCKLRRK2
SCHEMBL14982743 0.84 LRRK2 (0.84) EGFRKDRRETLCKLRRK2
SCHEMBL18158179 0.83 EGFR (0.79) EGFRKDRRETLCKPIK3CD
Hydrochloric Acid SCHEMBL8810155 0.82 EGFR (0.79) EGFRKDRRETLCKPIK3CD
Hydrochloric Acid SCHEMBL8811415 0.82 EGFR (0.79) EGFRKDRRETLCKPIK3CD
SCHEMBL1387182 0.82 EGFR (0.94) EGFRKDRRETLCKRIPK2
SCHEMBL29515328 0.82 EGFR (1.00) EGFRKDRRETLCKRIPK2
SCHEMBL1257431 0.82 EGFR (1.00) EGFRKDRRETLCKRIPK2
SCHEMBL8306414 0.81 LRRK2 (0.82) EGFRKDRRETLCKLRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0782570-A1 SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE IN MEDICINE THE WELLCOME FOUNDATION LIMITED (GB) 1997-07-09 EP disclosed
WO-1996009294-A1 SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE IN MEDICINE THE WELLCOME FOUNDATION LIMITED (GB) 1996-03-28 WO disclosed