SCHEMBL8808277

SCHEMBL8808277

Cc1ccc(C(C)N(O)C(=O)Nc2ccccc2)o1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 4/20 0.57
MTOR P42345 1/20 0.49
HPGD P15428 4/20 0.44
RAB9A P51151 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
NPC1 O15118 2/20 0.42
TSHR P16473 1/20 0.41
MAPT P10636 3/20 0.41
LMNA P02545 2/20 0.41
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
ALDH1A1 P00352 4/20 0.40
KLK7 P49862 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
ALOX15 P16050 1/20 0.39
HSD17B10 Q99714 1/20 0.39
KDM4E B2RXH2 1/20 0.39
PKM P14618 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8806331 0.80 ALOX5 (0.66) ALOX5HPGDALDH1A1KLK7
SCHEMBL8805696 0.80 RAB9A (0.56) ALOX5RAB9ASMN1; SMN2NPC1TSHR
SCHEMBL7608931 0.76 MTOR (0.57) MTORHPGDRAB9ASMN1; SMN2NPC1
SCHEMBL8807791 0.73 ALOX5 (1.00) ALOX5
Ammonia Solution, Strong SCHEMBL8807165 0.72 ALOX5 (0.97) ALOX5
SCHEMBL8806921 0.72 ALOX5 (0.97) ALOX5
SCHEMBL23200035 0.71 TSHR (0.53) ALOX5MTORHPGDTSHRMAPT
SCHEMBL7611785 0.71 NPY5R (0.57) MTORHPGDRAB9ASMN1; SMN2NPC1
SCHEMBL7610023 0.70 MEN1 (0.51) MTORHPGDRAB9ASMN1; SMN2NPC1
SCHEMBL9831966 0.69 MAPT (0.48) ALOX5HPGDRAB9ASMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0320628-B1 Substituted furan compounds which are useful in inhibiting lipoxygenase enzymes, particularly 5-lipoxygenase ABBOTT LAB (US) 1997-01-15 EP disclosed
US-5112848-A Antiasthmatics and antiarthritic agents ABBOTT LABORATORIES (US) 1992-05-12 US disclosed
EP-0388429-A4 FURAN AND PYRROLE CONTAINING LIPOXYGENASE INHIBITING COMPOUNDS 1991-08-21 EP disclosed
EP-0388429-A1 FURAN AND PYRROLE CONTAINING LIPOXYGENASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1990-09-26 EP disclosed
EP-0320628-A1 Substituted furan compounds which are useful in inhibiting lipoxygenase enzymes, particularly 5-lipoxygenase ABBOTT LABORATORIES (US) 1989-06-21 EP disclosed
WO-1989004299-A1 FURAN AND PYRROLE CONTAINING LIPOXYGENASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1989-05-18 WO disclosed