SCHEMBL8808557

SCHEMBL8808557

CC/C(O)=C(\C#N)C(=O)Nc1ccc(C(=O)c2ccc(Br)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
HPGD P15428 1/20 0.46
RAB9A P51151 1/20 0.46
DHODH Q02127 5/20 0.45
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
MAPT P10636 3/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
GAA P10253 1/20 0.42
CYP2C9 P11712 1/20 0.42
PKM P14618 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
LMNA P02545 1/20 0.42
THRB P10828 1/20 0.42
BLM P54132 1/20 0.42
BTK Q06187 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
PLK3 Q9H4B4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9080497 1.00 ALDH1A1 (0.46) ALDH1A1HPGDRAB9ADHODHMEN1
SCHEMBL9079756 0.87 TP53 (0.48) ALDH1A1HPGDRAB9ADHODHMEN1
SCHEMBL8812638 0.87 MEN1 (0.54) ALDH1A1HPGDRAB9ADHODHMEN1
SCHEMBL8808540 0.87 TP53 (0.48) ALDH1A1HPGDRAB9ADHODHMEN1
SCHEMBL9079574 0.87 MEN1 (0.54) ALDH1A1HPGDRAB9ADHODHMEN1
SCHEMBL9080385 0.85 DHODH (0.62) ALDH1A1RAB9ADHODHMEN1KMT2A
SCHEMBL8810683 0.85 DHODH (0.62) ALDH1A1RAB9ADHODHMEN1KMT2A
SCHEMBL9081774 0.80 TP53 (0.54) ALDH1A1RAB9ADHODHMEN1KMT2A
SCHEMBL8811773 0.80 TP53 (0.54) ALDH1A1RAB9ADHODHMEN1KMT2A
SCHEMBL5914890 0.78 DHODH (0.70) ALDH1A1RAB9ADHODHMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0527736-B1 ISOXAZOLE-4-CARBOXAMIDES AND HYDROXYALKYLIDENE-CYANOACETAMIDES, DRUGS CONTAINING THESE COMPOUNDS AND USE OF SUCH DRUGS HOECHST AG (DE) 1997-04-16 EP disclosed
US-5532259-A ANTITUMOR HOECHST AKTIENGESELLSCHAFT (DE) 1996-07-02 US disclosed
US-5494911-A TREATING LEUKEMIA, SARCOMA, CARCINOMA, LYMPHOMA, SKIN CANCER HOECHST AKTIENGESELLSCHAFT (DE) 1996-02-27 US disclosed
WO-1991017748-A1 ISOXAZOLE-4-CARBOXAMIDES AND HYDROXYALKYLIDENE-CYANOACETAMIDES, DRUGS CONTAINING THESE COMPOUNDS AND USE OF SUCH DRUGS HOECHST AKTIENGESELLSCHAFT (DE) 1991-11-28 WO disclosed