SCHEMBL8808941

SCHEMBL8808941

COc1cccc2c1CCC[C@H]2CN(C)CCc1ccc2c(c1)CCC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.75
SLC6A4 P31645 3/20 0.75
ADRA2A P08913 1/20 0.70
ADRA2B P18089 1/20 0.70
ADRA2C P18825 1/20 0.70
DRD4 P21917 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8808946 1.00 HTR1A (0.75) HTR1ASLC6A4ADRA2AADRA2BADRA2C
SCHEMBL9325431 0.94 HTR1A (0.67) HTR1ASLC6A4
SCHEMBL9325424 0.94 HTR1A (0.67) HTR1ASLC6A4
SCHEMBL9326949 0.91 SLC6A4 (0.72) HTR1ASLC6A4ADRA2AADRA2BADRA2C
SCHEMBL8814536 0.91 SLC6A4 (0.72) HTR1ASLC6A4ADRA2AADRA2BADRA2C
SCHEMBL8812106 0.89 HTR1A (0.71) HTR1ASLC6A4
SCHEMBL8815142 0.89 SLC6A4 (0.71) HTR1ASLC6A4ADRA2AADRA2BADRA2C
SCHEMBL8812113 0.89 HTR1A (0.71) HTR1ASLC6A4
SCHEMBL8811506 0.89 HTR1A (0.68) HTR1ASLC6A4
SCHEMBL8809960 0.89 SLC6A4 (0.69) HTR1ASLC6A4ADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0646112-A4 TERTIARY AND SECONDARY AMINES AS ALPHA-2 ANTAGONISTS AND SEROTONIN UPTAKE INHIBITORS. ABBOTT LAB (US) 1997-04-02 EP claimed
EP-0646112-A1 TERTIARY AND SECONDARY AMINES AS ALPHA-2 ANTAGONISTS AND SEROTONIN UPTAKE INHIBITORS ABBOTT LABORATORIES (US) 1995-04-05 EP claimed
WO-1993012754-A2 TERTIARY AND SECONDARY AMINES AS ALPHA-2 ANTAGONISTS AND SEROTONIN UPTAKE INHIBITORS ABBOTT LABORATORIES (US) 1993-07-08 WO claimed
EP-0646112-A4 TERTIARY AND SECONDARY AMINES AS ALPHA-2 ANTAGONISTS AND SEROTONIN UPTAKE INHIBITORS. ABBOTT LAB (US) 1997-04-02 EP disclosed
EP-0646112-A1 TERTIARY AND SECONDARY AMINES AS ALPHA-2 ANTAGONISTS AND SEROTONIN UPTAKE INHIBITORS ABBOTT LABORATORIES (US) 1995-04-05 EP disclosed
US-5288749-A Treating central nervous system or cardiovascular disorders ABBOTT LABORATORIES (US) 1994-02-22 US disclosed
WO-1993012754-A2 TERTIARY AND SECONDARY AMINES AS ALPHA-2 ANTAGONISTS AND SEROTONIN UPTAKE INHIBITORS ABBOTT LABORATORIES (US) 1993-07-08 WO disclosed