SCHEMBL8809186

SCHEMBL8809186

COc1cc2c(cc1OC)CN(CCCOc1ccc(NC(=O)c3ccc4ccccc4c3)cc1)CC2

nearest known ligand 0.78

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 16/20 0.78
ABCB1 P08183 14/20 0.78
DRD2 P14416 1/20 0.64
DRD1 P21728 1/20 0.64
DRD4 P21917 1/20 0.64
DRD3 P35462 1/20 0.64
MAOA P21397 1/20 0.58
MAOB P27338 1/20 0.58
CYP1A2 P05177 1/20 0.57
CYP2C8 P10632 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C9 P11712 1/20 0.57
ABCC1 P33527 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8808167 0.89 ABCG2 (0.88) ABCG2ABCB1DRD2DRD1DRD4
SCHEMBL8808324 0.88 ABCB1 (0.65) ABCG2ABCB1MAOAMAOB
SCHEMBL8812802 0.88 ABCG2 (1.00) ABCG2ABCB1
SCHEMBL8807711 0.84 ABCB1 (0.59) ABCG2ABCB1MAOAMAOB
SCHEMBL8807296 0.83 ABCG2 (0.79) ABCG2ABCB1MAOAMAOBCYP1A2
SCHEMBL14722808 0.83 DRD3 (0.90) ABCG2ABCB1DRD2DRD1DRD4
SCHEMBL8809580 0.82 ABCB1 (0.59) ABCG2ABCB1DRD1DRD4DRD3
SCHEMBL8809233 0.81 ABCG2 (0.78) ABCG2ABCB1MAOBCYP1A2CYP2C8
SCHEMBL8809520 0.80 ABCB1 (0.55) ABCG2ABCB1MAOAMAOB
SCHEMBL4040694 0.80 ABCB1 (0.77) ABCG2ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5663179-A CAN SENSITIZE MULTIDRUG RESISTANT CANCER CELLS TO CHEMOTHERAPEUTIC AGENTS LABORATOIRES GLAXO SA (FR) 1997-09-02 US disclosed
EP-0649410-B1 ANILIDE DERIVATIVES GLAXO LAB SA (FR) 1997-05-02 EP disclosed