SCHEMBL8809202

SCHEMBL8809202

CCCCc1nc(CC(C(=O)N[C@@H](Cc2cccc3ccccc23)C(=O)OCc2ccccc2)c2ccc3c(c2)OCO3)c(C(=O)OC(C)(C)C)[nH]1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 7/20 0.40
TACR1 P25103 2/20 0.38
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
IL1RN P18510 1/20 0.35
ERAP2 Q6P179 1/20 0.35
ACE P12821 1/20 0.35
ALDH1A1 P00352 2/20 0.35
LMNA P02545 2/20 0.35
MAPT P10636 1/20 0.35
CYP3A4 P08684 3/20 0.34
REN P00797 1/20 0.34
POLB P06746 1/20 0.34
MAPK1 P28482 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8809374 0.93 EDNRA (0.40) EDNRACTSSCTSKACEALDH1A1
SCHEMBL8809473 0.91 TACR1 (0.45) TACR1IL1RNERAP2MAPK1
SCHEMBL8807936 0.89 TACR1 (0.45) TACR1IL1RNERAP2MAPK1
SCHEMBL8809339 0.88 EDNRA (0.44) EDNRAACEALDH1A1LMNAMAPT
SCHEMBL8810904 0.87 TACR1 (0.46) TACR1IL1RNERAP2MAPK1
SCHEMBL8809082 0.86 EDNRA (0.44) EDNRAACEALDH1A1LMNAMAPT
SCHEMBL8807044 0.85 TACR1 (0.47) TACR1IL1RNERAP2ALDH1A1LMNA
SCHEMBL8807036 0.85 SMN1; SMN2 (0.43) EDNRATACR1CTSSCTSKLMNA
SCHEMBL8810295 0.84 MAPK1 (0.44) CTSSCTSKACEPOLBMAPK1
SCHEMBL8807991 0.83 MAPK1 (0.43) CTSSCTSKACEPOLBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0792265-A1 ENDOTHELIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-09-03 EP disclosed