SCHEMBL8809374

SCHEMBL8809374

CCCCc1nc(C[C@H](C(=O)N[C@@H](Cc2cccc3ccccc23)C(=O)O)c2ccc3c(c2)OCO3)c(C(=O)OC(C)(C)C)[nH]1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 5/20 0.40
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
MME P08473 1/20 0.38
ACE P12821 1/20 0.38
CPA1 P15085 1/20 0.38
ACE2 Q9BYF1 1/20 0.38
ALDH1A1 P00352 2/20 0.36
LMNA P02545 2/20 0.36
MAPT P10636 1/20 0.36
POLB P06746 1/20 0.35
MAPK1 P28482 1/20 0.35
HRH4 Q9H3N8 1/20 0.35
CYP3A4 P08684 3/20 0.34
PTGFR P43088 2/20 0.34
GAA P10253 1/20 0.34
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8809202 0.93 EDNRA (0.40) EDNRACTSSCTSKACEALDH1A1
SCHEMBL8810295 0.91 MAPK1 (0.44) CTSSCTSKACEPOLBMAPK1
SCHEMBL8807991 0.89 MAPK1 (0.43) CTSSCTSKACEPOLBMAPK1
SCHEMBL8807806 0.87 MAPK1 (0.45) CTSSCTSKACEPOLBMAPK1
SCHEMBL8807025 0.86 EDNRA (0.41) EDNRAMMEALDH1A1LMNAMAPT
SCHEMBL8807036 0.85 SMN1; SMN2 (0.43) EDNRACTSSCTSKLMNAMAPT
SCHEMBL8807746 0.84 MAPK1 (0.46) CTSSCTSKACEPOLBMAPK1
SCHEMBL8809473 0.84 TACR1 (0.45) MAPK1
SCHEMBL8809676 0.83 EDNRA (0.41) EDNRAMMEALDH1A1LMNAMAPT
SCHEMBL8807936 0.82 TACR1 (0.45) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0792265-A1 ENDOTHELIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-09-03 EP disclosed