SCHEMBL8809268

SCHEMBL8809268

Cc1ccc(-c2ccc(O)cc2)c(-c2ccc(OCCN3CCCCC3)cc2)n1

nearest known ligand 0.65

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 19/20 0.65
ESR2 Q92731 18/20 0.65
KDM4E B2RXH2 1/20 0.61
ALDH1A1 P00352 1/20 0.61
TP53 P04637 1/20 0.61
CYP1A2 P05177 1/20 0.61
CYP3A4 P08684 1/20 0.61
MAPT P10636 1/20 0.61
CYP2C9 P11712 1/20 0.61
ALOX15 P16050 1/20 0.61
TSHR P16473 1/20 0.61
HSD17B10 Q99714 1/20 0.61
TDP1 Q9NUW8 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8810633 0.99 ESR1 (0.65) ESR1ESR2KDM4EALDH1A1TP53
SCHEMBL8808818 0.91 LTA4H (0.55) ESR1ESR2KDM4EALDH1A1TP53
SCHEMBL8809840 0.90 LTA4H (0.56) ESR1ESR2KDM4EALDH1A1TP53
SCHEMBL8810978 0.86 ESR1 (0.66) ESR1ESR2KDM4EALDH1A1TP53
SCHEMBL8811463 0.83 ESR1 (0.61) ESR1ESR2KDM4EALDH1A1TP53
SCHEMBL8808018 0.82 ESR1 (0.61) ESR1ESR2KDM4EALDH1A1TP53
SCHEMBL8809777 0.80 CNR1 (0.56) ALDH1A1CYP1A2
SCHEMBL1359959 0.80 ESR1 (0.76) ESR1ESR2KDM4E
SCHEMBL699174 0.80 ESR1 (0.76) ESR1ESR2KDM4E
SCHEMBL2475993 0.78 ESR1 (0.75) ESR1ESR2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997004778-A1 PYRIDINE COMPOUNDS, INTERMEDIATES, PROCESSES, COMPOSITIONS, AND METHODS ELI LILLY AND COMPANY (US) 1997-02-13 WO disclosed