SCHEMBL8809840

SCHEMBL8809840

COc1ccc(-c2ccc(C)nc2-c2ccc(OCCN3CCCC3)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 3/20 0.56
MCHR1 Q99705 1/20 0.53
ESR1 P03372 8/20 0.53
ESR2 Q92731 4/20 0.52
HRH3 Q9Y5N1 3/20 0.50
MAPT P10636 2/20 0.49
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
TP53 P04637 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
ALOX15 P16050 1/20 0.49
TSHR P16473 1/20 0.49
HSD17B10 Q99714 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
KCNH2 Q12809 1/20 0.49
EBP Q15125 1/20 0.48
SIGMAR1 Q99720 1/20 0.48
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8808818 0.99 LTA4H (0.55) LTA4HMCHR1ESR1ESR2HRH3
SCHEMBL8810633 0.91 ESR1 (0.65) ESR1ESR2MAPTKDM4EALDH1A1
SCHEMBL8809777 0.90 CNR1 (0.56) HRH3ALDH1A1CYP1A2KCNH2SIGMAR1
SCHEMBL8809268 0.90 ESR1 (0.65) ESR1ESR2MAPTKDM4EALDH1A1
SCHEMBL8807859 0.88 LTA4H (0.56) LTA4HMCHR1ESR1ESR2HRH3
SCHEMBL8809238 0.84 LTA4H (0.58) LTA4HMCHR1ESR1HRH3KCNH2
SCHEMBL8810553 0.83 LTA4H (0.52) LTA4HMCHR1ESR1ESR2HRH3
SCHEMBL7443460 0.81 LTA4H (0.77) LTA4HMCHR1ESR1HRH3MAPT
SCHEMBL21121895 0.78 LTA4H (0.55) LTA4HMCHR1ESR1ESR2HRH3
SCHEMBL8809349 0.78 ESR1 (0.49) LTA4HMCHR1ESR1ESR2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997004778-A1 PYRIDINE COMPOUNDS, INTERMEDIATES, PROCESSES, COMPOSITIONS, AND METHODS ELI LILLY AND COMPANY (US) 1997-02-13 WO disclosed