SCHEMBL8809676

SCHEMBL8809676

CCCCCc1nc(CC(C(=O)O)c2ccc3c(c2)OCO3)c(C(=O)OC(C)(C)C)[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 3/20 0.41
AKR1C3 P42330 1/20 0.40
AKR1C2 P52895 1/20 0.40
MAPK9 P45984 1/20 0.39
TGFBR1 P36897 6/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.34
ALDH1A1 P00352 2/20 0.34
EDNRB P24530 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
KDM4E B2RXH2 1/20 0.34
TP53 P04637 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
MME P08473 1/20 0.34
OGA O60502 1/20 0.34
PTGFR P43088 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8807025 0.97 EDNRA (0.41) EDNRAAKR1C3AKR1C2MAPK9TGFBR1
SCHEMBL8807087 0.94 EDNRA (0.42) EDNRAAKR1C3AKR1C2MAPK9TGFBR1
SCHEMBL8809610 0.91 EDNRA (0.44) EDNRAAKR1C3AKR1C2MAPK9CYP1A2
SCHEMBL8809082 0.89 EDNRA (0.44) EDNRATGFBR1ALDH1A1LMNAMAPT
SCHEMBL8809339 0.87 EDNRA (0.44) EDNRATGFBR1ALDH1A1LMNAMAPT
SCHEMBL8810101 0.84 IL6ST (0.36) EDNRATGFBR1KMT2AALDH1A1EDNRB
SCHEMBL8807991 0.84 MAPK1 (0.43) KMT2ASMN1; SMN2
SCHEMBL8809374 0.83 EDNRA (0.40) EDNRAALDH1A1LMNAMAPTMME
SCHEMBL8811832 0.82 IL6ST (0.35) EDNRAALDH1A1EDNRBLMNAMAPT
SCHEMBL8807936 0.79 TACR1 (0.45) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0792265-A1 ENDOTHELIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-09-03 EP disclosed