SCHEMBL8809494

SCHEMBL8809494

c1ccc(COc2ccc(Sc3ncnc4ccccc34)cc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.57
ERBB2 P04626 4/20 0.57
CHEK2 O96017 1/20 0.57
ROS1 P08922 1/20 0.57
FLT3 P36888 1/20 0.57
ERBB4 Q15303 1/20 0.57
AURKB Q96GD4 1/20 0.57
CLK4 Q9HAZ1 1/20 0.57
MKNK2 Q9HBH9 1/20 0.57
ALDH1A1 P00352 1/20 0.54
HTT P42858 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
KDM1A O60341 2/20 0.45
STK17B O94768 1/20 0.44
LMNA P02545 4/20 0.44
CYP1A2 P05177 1/20 0.44
PTGS1 P23219 1/20 0.44
SLC6A2 P23975 1/20 0.44
CYP2C19 P33261 1/20 0.44
PTGS2 P35354 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8813070 0.82 KDM1A (0.66) EGFRERBB2FLT3HTTKDM1A
SCHEMBL27212829 0.81 KDM1A (0.58) EGFRERBB2AURKBCLK4ALDH1A1
SCHEMBL8810229 0.80 KDM1A (0.57) EGFRAURKBCLK4ALDH1A1HTT
SCHEMBL8811488 0.77 LMNA (0.71) EGFRERBB2CHEK2ROS1FLT3
SCHEMBL10337961 0.77 LMNA (0.64) LMNACYP1A2PTGS1SLC6A2CYP2C19
SCHEMBL1387173 0.76 EGFR (0.61) EGFRERBB2CHEK2ROS1FLT3
SCHEMBL6213388 0.75 MAPT (0.61) ALDH1A1HTTTDP1KDM1ALMNA
Benzylphenylether SCHEMBL8809498 0.74 EGFR (0.59) EGFRERBB2CHEK2ROS1FLT3
SCHEMBL4421697 0.73 MEN1 (0.49) EGFRERBB2CHEK2ROS1FLT3
SCHEMBL1387226 0.73 EGFR (1.00) EGFRERBB2CHEK2ROS1FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0782570-A1 SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE IN MEDICINE THE WELLCOME FOUNDATION LIMITED (GB) 1997-07-09 EP disclosed
WO-1996009294-A1 SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE IN MEDICINE THE WELLCOME FOUNDATION LIMITED (GB) 1996-03-28 WO disclosed