SCHEMBL8811488

SCHEMBL8811488

c1ccc(COc2ccc(COc3ncnc4ccccc34)cc2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.71
RAB9A P51151 3/20 0.63
L3MBTL1 Q9Y468 2/20 0.63
TSHR P16473 2/20 0.63
NPC1 O15118 1/20 0.63
EGFR P00533 3/20 0.63
ERBB2 P04626 3/20 0.63
CHEK2 O96017 1/20 0.63
ROS1 P08922 1/20 0.63
FLT3 P36888 1/20 0.63
ERBB4 Q15303 1/20 0.63
AURKB Q96GD4 1/20 0.63
CLK4 Q9HAZ1 1/20 0.63
MKNK2 Q9HBH9 1/20 0.63
CYP1A2 P05177 2/20 0.57
CYP2C19 P33261 2/20 0.57
CYP2C9 P11712 1/20 0.57
PDE5A O76074 1/20 0.52
RXFP1 Q9HBX9 1/20 0.50
MAOB P27338 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1387173 0.90 EGFR (0.61) LMNARAB9AL3MBTL1TSHRNPC1
SCHEMBL8810873 0.80 PDGFRB (0.68) LMNAEGFRERBB2FLT3ERBB4
SCHEMBL29244645 0.79 LMNA (0.68) LMNARAB9AL3MBTL1TSHRNPC1
SCHEMBL1680825 0.79 EGFR (0.76) LMNARAB9ATSHREGFRERBB2
Benzylphenylether SCHEMBL8809498 0.79 EGFR (0.59) LMNARAB9AL3MBTL1TSHRNPC1
SCHEMBL1387226 0.77 EGFR (1.00) RAB9ANPC1EGFRERBB2CHEK2
SCHEMBL8809494 0.77 EGFR (0.57) LMNARAB9AL3MBTL1TSHRNPC1
SCHEMBL14692125 0.77 LMNA (0.56) LMNARAB9AL3MBTL1TSHRNPC1
SCHEMBL8548739 0.76 RAB9A (0.69) LMNARAB9AL3MBTL1TSHRNPC1
Hydrochloric Acid SCHEMBL8810027 0.76 EGFR (0.97) RAB9ANPC1EGFRERBB2CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0782570-A1 SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE IN MEDICINE THE WELLCOME FOUNDATION LIMITED (GB) 1997-07-09 EP disclosed
WO-1996009294-A1 SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE IN MEDICINE THE WELLCOME FOUNDATION LIMITED (GB) 1996-03-28 WO disclosed