SCHEMBL8809659

SCHEMBL8809659

COc1cc(C(=N)N)ccc1CNC(=O)[C@@H]1CCCN1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.59
HTR2C P28335 9/20 0.54
HTR2B P41595 6/20 0.54
HTR2A P28223 4/20 0.54
GID4 Q8IVV7 1/20 0.47
HPGD P15428 1/20 0.43
HDAC1 Q13547 3/20 0.42
HDAC3 O15379 2/20 0.40
F2 P00734 1/20 0.40
QRFPR Q96P65 1/20 0.40
HDAC2 Q92769 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6483706 0.82 HTR2C (0.59) KDM4EHTR2CHTR2BHTR2AGID4
SCHEMBL6483702 0.82 HTR2C (0.59) KDM4EHTR2CHTR2BHTR2AGID4
Hydrochloric Acid SCHEMBL8377589 0.81 HTR2C (0.58) KDM4EHTR2CHTR2BHTR2AGID4
Hydrochloric Acid SCHEMBL7044040 0.81 HTR2C (0.58) KDM4EHTR2CHTR2BHTR2AGID4
SCHEMBL8809131 0.79 HTR2C (0.64) KDM4EHTR2CHTR2BHDAC1HDAC3
Hydrochloric Acid SCHEMBL5900833 0.78 HTR2C (0.62) KDM4EHTR2CHTR2BHDAC1HDAC3
Hydrochloric Acid SCHEMBL5900838 0.78 HTR2C (0.62) KDM4EHTR2CHTR2BHDAC1HDAC3
Trifluoroacetic Acid SCHEMBL18670028 0.76 KDM4E (0.55) KDM4EHTR2CHTR2BHTR2AGID4
Trifluoroacetic Acid SCHEMBL18670029 0.76 KDM4E (0.55) KDM4EHTR2CHTR2BHTR2AGID4
SCHEMBL8727237 0.75 PRSS1 (0.45) F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996025426-A9 NOVEL DIPEPTIDE AMIDINES AS THROMBIN INHIBITORS 1997-06-12 WO disclosed